The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jul. 28, 2026
Filed:
Sep. 16, 2022
Applicant:
Hoffmann-la Roche Inc., Little Falls, NJ (US);
Inventors:
Kirsten Andrea Graeser, Basel, CH;
Urs Schwitter, Reinach, CH;
Frank Stowasser, Basel, CH;
Florence Nicole Antoinette Tixeront, Kembs, FR;
Assignee:
Hoffmann-La Roche Inc., Little Falls, NJ (US);
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 413/12 (2006.01); A61K 31/5377 (2006.01); A61P 25/00 (2006.01); A61P 25/24 (2006.01);
U.S. Cl.
CPC ...
C07D 413/12 (2013.01); C07B 2200/13 (2013.01);
Abstract
Described herein are amorphous and crystalline forms of pharmaceutically acceptable salts of the TAAR1 agonist 5-ethyl-4-methyl-N-[4-[(2S) morpholin-2-yl]phenyl]-1H-pyrazole-3-carboxamide. Also described are pharmaceutical compositions suitable for administration to a mammal that include the TAAR1 agonist, and methods of using the TAAR1 agonist, alone and in combination with other compounds, for treating diseases or conditions that are associated with TAAR1 activity.