The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 10, 2026

Filed:

Aug. 06, 2020
Applicant:

Janssen Pharmaceutica NV, Beerse, BE;

Inventors:

Dominique Paul M Depre, Hamme-Mille, BE;

Kiran Matcha, Turnhout, BE;

Florian Damien Medina, Brussels, BE;

Pieter Westerduin, Lichtaart, BE;

Cheng Yi Chen, San Diego, CA (US);

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 487/04 (2006.01); C07C 249/16 (2006.01); C07C 251/76 (2006.01); C07C 251/78 (2006.01); C07D 249/06 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); C07C 249/16 (2013.01); C07C 251/76 (2013.01); C07C 251/78 (2013.01); C07D 249/06 (2013.01);
Abstract

Processes for preparing (((3aR,6aS)-5-(4,6-dimethylpyrimidin-2-yl)hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)(2-fluoro-6-(2H-1,2,3-triazol-2-yl)phenyl)methanone are described, which are useful for commercial manufacturing. Said compound is an orexin receptor modulator and may be useful in pharmaceutical compositions and methods for the treatment of diseased states, disorders, and conditions mediated by orexin activity, such as insomnia and depression.


Find Patent Forward Citations

Depre, Dominique Paul M. (2026). Synthetic methods of making (2h-1, 2, 3-triazol-2-yl) phenyl compounds as orexin receptor modulators (U.S. Patent No. 12570658). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/12570658

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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