The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 02, 2025

Filed:

Aug. 15, 2022
Applicant:

Chinese Academy of Medical Sciences Institute of Medicinal Plant Development, Beijing, CN;

Inventors:

Xiaobo Sun, Beijing, CN;

Yu Tian, Beijing, CN;

Xiao Sun, Beijing, CN;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/24 (2006.01); A61K 31/235 (2006.01); A61P 9/10 (2006.01); C07C 68/00 (2020.01); C07C 69/76 (2006.01); C07C 205/59 (2006.01);
U.S. Cl.
CPC ...
A61K 31/24 (2013.01); A61K 31/235 (2013.01); A61P 9/10 (2018.01); C07C 68/00 (2013.01); C07C 69/76 (2013.01); C07C 205/59 (2013.01);
Abstract

Disclosed are a hydroxypentyl benzoic acid diester compound, a method preparing the same, and an application of the same. This application uses a combination principle, on the one hand, the medicine concentration of butylphthalide in cerebral vessels is improved through a function of promoting the medicine to penetrate through a blood-brain barrier of dexborneol, and a multi-target multi-channel synergistic brain protection effect of the medicine is exerted; on the other hand, the treatment effect of dexborneol on cerebral ischemia is exerted. Anti-cerebral ischemia in-vivo pharmacodynamic activity evaluation is carried out on the synthesized compound, a high-activity candidate medicine is obtained, and industrial production can be achieved through the synthesis method.


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