The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jul. 29, 2025
Filed:
Sep. 27, 2019
Richter Gedeon Nyrt., Budapest, HU;
György Szabó, Budapest, HU;
György István Túrós, Budapest, HU;
Olivér Éliás, Marcali, HU;
Benedek Imre Károlyi, Budapest, HU;
Péter Erdélyi, Budapest, HU;
Gábor Kapus, Pécel, HU;
RICHTER GEDEON NYRT., Budapest, HU;
Abstract
The present invention provides compounds of formula (I) and/or salt thereof and/or geometric isomer thereof and/or stereoisomer thereof and/or enantiomer thereof and/or racemate thereof and/or diastereomer thereof and/or biologically active metabolite thereof and/or prodrug thereof and/or solvate thereof and/or hydrate thereof and/or polymorph thereof having affinity and selectivity for the gamma-aminobutyric acid A receptor subunit alpha 5 and act as GABAα5 negative allosteric modulators, thereby useful in the treatment or prevention of diseases related to the GABAα5 receptor, process for the preparation thereof, pharmaceutical compositions comprising them alone or in combination with one or more other active ingredients and their use as medicaments.