The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 10, 2024

Filed:

May. 16, 2019
Applicant:

Novartis Ag, Basel, CH;

Inventors:

Nicole Bieri, Muttenz, CH;

Andreas Kordikowski, Binningen, CH;

Bin Li, Changshu, CN;

Philipp Lustenberger, Allschwil, CH;

Rita Ramos, Allschwil, CH;

Vijay Sethuraman, Fremont, CA (US);

Sisi Zhang, Changshu, CN;

Assignee:

Novartis AG, Basel, CH;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 31/4162 (2006.01); A61K 31/5377 (2006.01); A61K 45/06 (2006.01); C07D 231/00 (2006.01); C07D 519/00 (2006.01); A61K 31/437 (2006.01); C07D 265/30 (2006.01); C07D 487/04 (2006.01);
U.S. Cl.
CPC ...
C07D 519/00 (2013.01); A61K 31/4162 (2013.01); A61K 31/5377 (2013.01); A61K 45/06 (2013.01); C07D 231/00 (2013.01); A61K 31/437 (2013.01); C07B 2200/13 (2013.01); C07D 265/30 (2013.01); C07D 487/04 (2013.01);
Abstract

This application relates to various crystalline forms of (S)—N-(4-((5-(1,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-4-yl)-3-methyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-1-yl)methyl)bicyclo[2.2.2]octan-1-yl)morpholine-3-carboxamide in its free form, as well as compositions, method of making and methods of using the same. In some embodiments the crystalline forms also contain water ('hydrates'). These materials are useful in the treatment of various autoimmune diseases, including systemic lupus erythematosus, cutaneous lupus, discoid lupus, mixed connective tissue disease, primary biliary cirrhosis, immune thrombocytopenia purpura, hidradenitis suppurativa, dermatomyositis, polymyositis, Sjögren's syndrome, arthritis, rheumatoid arthritis and psoriasis.


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