The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 30, 2024

Filed:

Mar. 09, 2022
Applicant:

Janssen Pharmaceutica NV, Beerse, BE;

Inventors:

Tongfei Wu, Boortmeerbeek, BE;

Dirk Brehmer, Freiburg, BE;

Lijs Beke, Antwerp, BE;

An Boeckx, Herentals, BE;

Gaston Stanislas Marcella Diels, Turnhout, BE;

Ronaldus Arnodus Hendrika Joseph Gilissen, Kasterlee, BE;

Edward Charles Lawson, Pipersville, PA (US);

Vineet Pande, Vosselaar, BE;

Marcus Cornelis Bernardus Catharina Paradé, Eindhoven, NL;

Wim Bert Griet Schepens, Sint Katelijne Waver, BE;

Johannes Wilhelmus John F. Thuring, Antwerp, BE;

Marcel Viellevoye, Breda, NL;

Weimei Sun, Lower Gwynedd, PA (US);

Lieven Meerpoel, Beerse, BE;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A01N 43/04 (2006.01); A61K 31/70 (2006.01); A61K 31/7076 (2006.01); A61K 31/519 (2006.01); A61K 31/53 (2006.01); C07D 471/04 (2006.01); A61P 35/00 (2006.01); A61K 31/5025 (2006.01);
U.S. Cl.
CPC ...
A61K 31/7076 (2013.01); A61K 31/5025 (2013.01); A61K 31/519 (2013.01); A61K 31/53 (2013.01); A61P 35/00 (2018.01); C07D 471/04 (2013.01);
Abstract

The present invention relates novel 6-6 bicyclic aromatic ring substituted nucleoside analogues of Formula (I) wherein the variables have the meaning defined in the claims. The compounds according to the present invention are useful as PRMT5 inhibitors. The invention further relates to pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as a medicament.


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