The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 24, 2023

Filed:

Feb. 26, 2021
Applicant:

Insmed Incorporated, Bridgewater, NJ (US);

Inventors:

Vladimir Malinin, Plainsboro, NJ (US);

Walter Perkins, Neshanic Station, NJ (US);

Franziska Leifer, Princeton, NJ (US);

Donna Konicek, Belle Mead, NJ (US);

Zhili Li, Kendall Park, NJ (US);

Adam Plaunt, Phillipsburg, NJ (US);

Assignee:

Insmed Incorporated, Bridgewater, NJ (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 69/734 (2006.01); C07C 69/712 (2006.01); A61K 47/60 (2017.01); A61K 47/54 (2017.01); C07C 69/736 (2006.01); C07C 69/753 (2006.01); C07C 235/22 (2006.01); C07C 235/20 (2006.01); A61K 31/165 (2006.01); A61K 31/216 (2006.01); A61K 31/225 (2006.01); A61K 47/06 (2006.01); A61K 9/00 (2006.01); A61P 9/12 (2006.01); A61P 11/00 (2006.01); A61K 9/10 (2006.01); A61K 9/14 (2006.01); A61K 9/51 (2006.01); A61K 47/14 (2017.01); A61K 47/24 (2006.01); A61K 47/28 (2006.01); A61K 47/34 (2017.01); A61M 15/00 (2006.01); A61M 16/14 (2006.01);
U.S. Cl.
CPC ...
C07C 69/734 (2013.01); A61K 9/0019 (2013.01); A61K 9/0043 (2013.01); A61K 9/0053 (2013.01); A61K 9/0073 (2013.01); A61K 9/0075 (2013.01); A61K 9/0078 (2013.01); A61K 9/10 (2013.01); A61K 9/14 (2013.01); A61K 9/51 (2013.01); A61K 31/165 (2013.01); A61K 31/216 (2013.01); A61K 31/225 (2013.01); A61K 47/06 (2013.01); A61K 47/14 (2013.01); A61K 47/24 (2013.01); A61K 47/28 (2013.01); A61K 47/34 (2013.01); A61K 47/543 (2017.08); A61K 47/544 (2017.08); A61K 47/60 (2017.08); A61M 15/009 (2013.01); A61M 15/0085 (2013.01); A61M 16/14 (2013.01); A61P 9/12 (2018.01); A61P 11/00 (2018.01); C07C 69/712 (2013.01); C07C 69/736 (2013.01); C07C 69/753 (2013.01); C07C 235/20 (2013.01); C07C 235/22 (2013.01); A61M 2202/064 (2013.01); C07C 2601/18 (2017.05); C07C 2603/14 (2017.05);
Abstract

Prostacyclin compounds and compositions comprising the same are provided herein. Specifically, prostacyclin compounds comprising treprostinil covalently linked to a linear C-Calkyl, branched C-Calkyl, linear C-Calkenyl, branched C-Calkenyl, aryl, aryl-C-Calkyl or an amino acid or a peptide (e.g., dipeptide, tripeptide, tetrapeptide) are described. The linkage, in one embodiment, is via a carbamate, amide or ester bond. Prostacyclin compounds provided herein can also include at least one hydrogen atom substituted with at least one deuterium atom. Methods for treating pulmonary hypertension (e.g., pulmonary arterial hypertension) and portopulmonary hypertension are also provided.


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