The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 13, 2022

Filed:

Oct. 30, 2020
Applicant:

Mosaic Biosciences, Inc., Boulder, CO (US);

Inventors:

Alexei V. Kazantsev, Erie, CO (US);

Peter D. Mariner, Superior, CO (US);

Martin Stanton, Boulder, CO (US);

Assignee:

Mosaic Biosciences, Inc., Boulder, CO (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 47/60 (2017.01); C08G 75/12 (2016.01); C08G 75/045 (2016.01); C08J 3/24 (2006.01); C08G 81/00 (2006.01); C08H 1/00 (2006.01); C07K 1/107 (2006.01); C12N 9/36 (2006.01); C08B 37/00 (2006.01); C07K 14/78 (2006.01); C08J 3/075 (2006.01); C08L 101/16 (2006.01); A61K 9/06 (2006.01); A61K 38/08 (2019.01); A61K 38/10 (2006.01); A61K 38/39 (2006.01); C08G 65/334 (2006.01);
U.S. Cl.
CPC ...
A61K 47/60 (2017.08); A61K 9/06 (2013.01); A61K 38/08 (2013.01); A61K 38/10 (2013.01); A61K 38/39 (2013.01); C07K 1/1077 (2013.01); C07K 14/78 (2013.01); C08B 37/0069 (2013.01); C08B 37/0075 (2013.01); C08G 65/3342 (2013.01); C08G 75/045 (2013.01); C08G 75/12 (2013.01); C08G 81/00 (2013.01); C08H 1/00 (2013.01); C08J 3/075 (2013.01); C08J 3/246 (2013.01); C08L 101/16 (2013.01); C12N 9/2462 (2013.01); C12Y 302/01017 (2013.01); C08G 2210/00 (2013.01); C08G 2650/04 (2013.01); C08G 2650/16 (2013.01); C08G 2650/20 (2013.01); C08J 2300/16 (2013.01); C08J 2371/02 (2013.01); C08J 2389/00 (2013.01);
Abstract

Provided are methods for linking polypeptides (including peptides and proteins) to other moieties using radical imitated thiol-ene chemistries, for example, modifying a polypeptide by introducing reactive thiol groups and reacting the thiol groups with olefin-containing reagents or alkyne-containing reagents under conditions that support radical thiol-ene or thiol-yne reactions. The reactive thiol groups have greater activity for radical thiol-ene reactions that a cysteine thiol group, including thiol groups that are separated from the peptide backbone by at least two carbon atoms, for example, the thiol group of a homocysteine residue. Also provided are compositions and biomaterials containing the linked polypeptides, for example, peptide and protein conjugates, and thiol-ene based biocompatible hydrogel polymers, and their uses in the medical field.


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