The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Aug. 02, 2022
Filed:
Jan. 13, 2020
Applicant:
Lupin Inc., Baltimore, MD (US);
Inventors:
Assignee:
Lupin, Inc., Baltimore, MD (US);
Primary Examiner:
Int. Cl.
CPC ...
C07D 239/46 (2006.01); A61K 31/513 (2006.01); A61P 15/00 (2006.01); A61P 29/00 (2006.01);
U.S. Cl.
CPC ...
A61K 31/513 (2013.01); A61P 15/00 (2018.01); A61P 29/00 (2018.01);
Abstract
New deuterated analogs of elagolix are provided. The novel deuterated elagolix analogs differ from the only previously disclosed deuterated elagolix analogs in structure based on the exclusion of deuterium at certain sites in the compounds and the inclusion of deuterium at other sites. Also provided are new formulations for deuterated elagolix compounds and methods of using such compounds and formulations in the modification of mammalian physiology and especially in the treatment and prevention of a number of diseases and disorders, including endometriosis-associated pain and uterine fibroid conditions.