The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 19, 2022

Filed:

Nov. 20, 2018
Applicant:

Purdue Research Foundation, West Lafayette, IN (US);

Inventors:

Mingji Dai, West Lafayette, IN (US);

Ji-Xin Cheng, Newton, MA (US);

Assignee:

Purdue Research Foundation, West Lafayette, IN (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07J 9/00 (2006.01); G01N 33/52 (2006.01); C07J 17/00 (2006.01); C07J 41/00 (2006.01);
U.S. Cl.
CPC ...
C07J 9/00 (2013.01); C07J 9/005 (2013.01); C07J 17/00 (2013.01); C07J 41/0094 (2013.01); G01N 33/52 (2013.01);
Abstract

A method of forming a probe, wherein the method includes converting cholenic acid into a compound with a terminal alkyne group, wherein the converting the cholenic acid comprises using a sequence, wherein the sequence comprises synthesizing a THP-protection group, LiAlH4 reduction, Dess-Martin oxidation, and Seyferth-Gilbert-Bestmann homologation. The method additionally includes forming A-Chol by removing the THP-protection. Further, the method includes forming PhA-Chol from the compound with the terminal alkyne group via a palladiumcatalyzed Sonogashira reaction. Additionally, the method includes forming PhDY Chol from the compound with the terminal alkyne group via a coppercatalyzed Cadiot-Chodkiewicz reaction.


Find Patent Forward Citations

Loading…