The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 24, 2022

Filed:

Mar. 25, 2019
Applicant:

The Board of Trustees of the Leland Stanford Junior University, Stanford, CA (US);

Inventors:

Isabella A. Graef, Woodside, CA (US);

Mamoun M. Alhamadsheh, Fremont, CA (US);

Assignee:

Other;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/12 (2006.01); C07D 231/12 (2006.01); A61K 31/4196 (2006.01); A61K 31/428 (2006.01); A61K 31/433 (2006.01); C07D 487/04 (2006.01); A61K 31/519 (2006.01); A61K 31/166 (2006.01); G01N 21/64 (2006.01);
U.S. Cl.
CPC ...
A61K 31/12 (2013.01); A61K 31/166 (2013.01); A61K 31/4196 (2013.01); A61K 31/428 (2013.01); A61K 31/433 (2013.01); A61K 31/519 (2013.01); C07D 231/12 (2013.01); C07D 487/04 (2013.01); G01N 21/6428 (2013.01);
Abstract

Disclosed herein are compounds and compositions thereof which find use in increasing stability of TTR tetramers reducing its tendency to misfold and form aggregates. Also provided herein are methods for using these compounds and compositions for increasing stability of TTR and thereby decreasing aggregate formation by TTR. Also disclosed herein are methods to screen for candidate compounds that increase stability of TTR. Also disclosed herein are heterobifunctional compounds that include a TTR binding compound connected to a targeting moiety via a linker, for use in disrupting PPIs of a target protein.


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