The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 10, 2022

Filed:

Aug. 01, 2012
Applicants:

Varghese John, San Francisco, CA (US);

Dale E. Bredesen, Novato, CA (US);

Inventors:

Varghese John, San Francisco, CA (US);

Dale E. Bredesen, Novato, CA (US);

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 453/02 (2006.01); C07D 451/12 (2006.01); A61K 31/439 (2006.01); A61K 31/444 (2006.01); A61K 45/06 (2006.01);
U.S. Cl.
CPC ...
C07D 453/02 (2013.01); A61K 31/439 (2013.01); A61K 31/444 (2013.01); A61K 45/06 (2013.01); C07D 451/12 (2013.01);
Abstract

In various embodiments, compositions and methods are provided for treatment and/or prevention of amyloidogenic diseases. In certain embodiments, the methods entail administering an effective amount of a tropinol ester to a subject in need thereof for prophylactic or therapeutic effect. The methods are particularly useful for prophylactic and therapeutic treatment of Alzheimer's disease. In certain embodiments, methods of reducing the risk, lessening the severity, or delaying the progression or onset of a disease characterized by beta-amyloid deposits in the brain of a mammal are also provided. In certain embodiments, methods of directly or indirectly inhibiting the C-terminal cleavage of APP resulting in the formation of APP-C31 peptide and APPneo (AP-P664) in a mammal are provided.


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