The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 21, 2021

Filed:

Sep. 27, 2017
Applicant:

Beigene, Ltd., Grand Cayman, KY;

Inventors:

Lai Wang, Beijing, CN;

Zhiyu Tang, Beijing, CN;

Lusong Luo, Beijing, CN;

Min Wei, Beijing, CN;

Kang Li, Beijing, CN;

Jing Song, Beijing, CN;

Tong Zhang, Beijing, CN;

Hexiang Wang, Beijing, CN;

Bo Ren, Beijing, CN;

Changyou Zhou, Princeton, NJ (US);

Assignee:

BEIGENE, LTD., Grand Cayman, KY;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/551 (2006.01); A61K 45/00 (2006.01); A61P 35/00 (2006.01); C07D 471/16 (2006.01); C07D 487/06 (2006.01); C07D 487/16 (2006.01); A61K 31/282 (2006.01); A61K 31/337 (2006.01); A61K 31/357 (2006.01); A61K 39/395 (2006.01); C07K 16/28 (2006.01);
U.S. Cl.
CPC ...
A61K 31/551 (2013.01); A61K 31/282 (2013.01); A61K 31/337 (2013.01); A61K 31/357 (2013.01); A61K 39/3955 (2013.01); A61P 35/00 (2018.01); C07K 16/2818 (2013.01);
Abstract

Disclosed herein is a method for the prevention, delay of progression or treatment of cancer in a subject, comprising administering to the subject in need thereof a PARP inhibitor, particularly, (R)-2-fluoro-10a-methyl-7,8,9,10,10a,11-hexahydro-5,6,7a,11-tetraazacyclohepta[def]cyclopenta[a]fluoren-4(5H)-one, a sesqui-hydrate thereof, or a pharmaceutically acceptable salt thereof, in combination with an immune checkpoint inhibitor or a chemotherapeutic agent. Also, disclosed a pharmaceutical combination comprising a PARP inhibitor, particularly, (R)-2-fluoro-10a-methyl-7,8,9,10,10a,11-hexahydro-5,6,7a,11-tetraazacyclohepta[def]cyclopenta[a]fluoren-4(5H)-one, a sesqui-hydrate thereof, or a pharmaceutically acceptable salt thereof, in combination with an immune checkpoint inhibitor, or a chemotherapeutic agent and the use thereof.


Find Patent Forward Citations

Loading…