The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 30, 2021

Filed:

Jun. 03, 2020
Applicant:

Wisconsin Alumni Research Foundation, Madison, WI (US);

Inventors:

Jamey Weichert, Sun Prairie, WI (US);

Anatoly Pinchuk, Fitchburg, WI (US);

Reinier Hernandez, Madison, WI (US);

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 51/00 (2006.01); A61M 36/14 (2006.01); C07F 9/6524 (2006.01); C07B 59/00 (2006.01); G01N 33/574 (2006.01); A61K 51/04 (2006.01); A61N 5/10 (2006.01); G01N 33/60 (2006.01);
U.S. Cl.
CPC ...
C07F 9/6524 (2013.01); A61K 51/0482 (2013.01); A61K 51/0489 (2013.01); A61N 5/10 (2013.01); C07B 59/004 (2013.01); G01N 33/574 (2013.01); G01N 33/60 (2013.01);
Abstract

Alkylphosphocholine analogs incorporating a chelating moiety that chelates a radioactive metal isotope are disclosed herein. The alkylphophocholine analogs, which can be used to treat or detect solid tumors, have the formula: Rincludes a chelating agent that is chelated to a metal atom, wherein the metal atom is a positron or single photon emitting metal isotope with a half life of greater than or equal to 4 hours, or an alpha, beta or Auger emitting metal isotope with a half life of greater than 6 hours and less than 30 days; a is 0 or 1; n is an integer from 12 to 30; m is 0 or 1; Y is —H, —OH, —COOH, —COOX, —OCOX, or —OX, wherein X is an alkyl or an arylalkyl; Ris —NH, —NHZ, —NHZ, or —NZ, wherein each Z is independently an alkyl or an aroalkyl; and b is 1 or 2.


Find Patent Forward Citations

Loading…