The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 23, 2021

Filed:

Mar. 29, 2017
Applicants:

University of Virginia Patent Foundation, Charlottesville, VA (US);

Virginia Tech Intellectual Properties, Inc., Blacksburg, VA (US);

Inventors:

Steven Brandon Thorpe, Palmyra, VA (US);

Webster L. Santos, Blacksburg, VA (US);

Kevin R. Lynch, Charlottesville, VA (US);

Assignees:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 403/14 (2006.01); C07D 403/04 (2006.01); C07D 413/14 (2006.01); C07D 413/04 (2006.01);
U.S. Cl.
CPC ...
C07D 413/14 (2013.01); C07D 413/04 (2013.01);
Abstract

Sphingosine kinases are enzymes that catalyze the biosynthesis of sphingosine-1-phosphate. The invention provides prodrugs of compounds that are effective for inhibition of sphingosine kinase type 1, sphingosine kinase type 2, or both, according to formula (I) as described herein. Formula I compounds are useful in the treatment of a range of diseases wherein increasing the level of sphingosine-1-phosphate in blood is medically indicated. The invention also provides pharmaceutical compositions of Formula I compounds.


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