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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 11111220 B1

PDFFull Text
Expired
Date of Patent:
Sep. 07, 2021

Filed:

Oct. 16, 2018

Propanamine derivatives for treating pain and pain related conditions

Applicant:

Esteve Pharmaceuticals, S.a., Barcelona, ES;

Inventors:

Carmen Almansa-Rosales, Barcelona, ES;

Félix Cuevas-Cordobés, Valdemoro, ES;

Assignee:

ESTEVE PHARMACEUTICALS, S.A., Barcelona, ES;

Attorney:

Hueschen and Sage

Primary Examiner:

Samantha L Shterengarts

Int. Cl.
CPC ...
A61K 31/505 (2006.01); C07D 239/48 (2006.01); C07C 235/56 (2006.01); C07D 211/58 (2006.01); C07D 213/75 (2006.01); C07D 213/82 (2006.01); C07D 239/34 (2006.01); C07D 333/20 (2006.01); C07D 409/12 (2006.01); C07D 413/12 (2006.01);
U.S. Cl.
CPC ...
C07D 239/48 (2013.01); C07C 235/56 (2013.01); C07D 211/58 (2013.01); C07D 213/75 (2013.01); C07D 213/82 (2013.01); C07D 239/34 (2013.01); C07D 333/20 (2013.01); C07D 409/12 (2013.01); C07D 413/12 (2013.01);
Abstract

The present invention relates to new compounds of formula (I) that show great affinity and activity towards the subunit α2δ of voltage-gated calcium channels (VGCC), especially the α2δ-1 subunit of voltage-gated calcium channels or dual activity towards the subunit α2δ of voltage-gated calcium channels (VGCC), especially the α2δ-1 subunit of voltage-gated calcium channels, and the noradrenaline transporter (NET). The invention is also related to the process for the preparation of said compounds as well as to compositions comprising them, and to their use as medicaments.

Find Patent Forward Citations

Almansa-Rosales, Carmen. (2021). Propanamine derivatives for treating pain and pain related conditions (U.S. Patent No. 11111220). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/11111220

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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