The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Aug. 10, 2021
Filed:
Aug. 19, 2019
Applicant:
Biohaven Therapeutics Ltd., New Haven, CT (US);
Inventor:
Anthony Marfat, Mystic, CT (US);
Assignee:
Biohaven Therapeutics Ltd., New Haven, CT (US);
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 277/82 (2006.01); A61K 31/428 (2006.01); A61K 9/14 (2006.01); C07D 417/12 (2006.01); C07F 9/6541 (2006.01); A61K 47/16 (2006.01);
U.S. Cl.
CPC ...
A61K 31/428 (2013.01); A61K 9/14 (2013.01); A61K 47/16 (2013.01); C07D 277/82 (2013.01); C07D 417/12 (2013.01); C07F 9/6541 (2013.01);
Abstract
Disclose are amine prodrugs and methods of synthesis thereof. In particular, the amine prodrug comprises a drug molecule and at least one or more prodrug appendage moieties and the method for synthesis the amine prodrug comprises a step of coupling the drug molecule and at least one or more prodrug appendage moieties. Also disclosed are exemplary riluzole prodrugs and methods of synthesis thereof.