The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 06, 2021

Filed:

Dec. 12, 2019
Applicant:

Kaohsiung Medical University, Kaohsiung, TW;

Inventors:

Yeh-Long Chen, Kaohsiung, TW;

Tian-Lu Cheng, Kaohsiung, TW;

Cherng-Chyi Tzeng, Kaohsiung, TW;

Chih-Hua Tseng, Kaohsiung, TW;

Ta-Chun Cheng, Kaohsiung, TW;

Kai-Wen Cheng, Kaohsiung, TW;

Wei-Fen Luo, Kaohsiung, TW;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/437 (2006.01); A61K 45/06 (2006.01); C07D 471/04 (2006.01); A61P 35/00 (2006.01); A61K 31/055 (2006.01); A61K 31/03 (2006.01);
U.S. Cl.
CPC ...
A61K 31/437 (2013.01); A61K 31/055 (2013.01); A61K 45/06 (2013.01); A61P 35/00 (2018.01); C07D 471/04 (2013.01); A61K 31/03 (2013.01);
Abstract

The present invention provides novel pyrazolo[4,3-c]quinoline derivatives exhibiting specifically inhibition activity to microbiota β-glucuronidase, whereby providing potent activities to prevent chemotherapy-induced diarrhea (CID) of cancers. Therefore, the compounds of the present invention can be used as (1) chemotherapy-adjuvant to prevent chemotherapy-induced diarrhea (CID) and enhance chemotherapeutic efficiency of cancers; (2) health-food supplement to prevent the carcinogens induced colon carcinoma.


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