The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 25, 2021

Filed:

Jan. 05, 2017
Applicants:

Universite Paris-sud, Orsay, FR;

Centre National DE LA Recherche Scientifique (Cnrs), Paris, FR;

Inventors:

Mouâd Alami, Bussy Saint Georges, FR;

Abdallah Hamze, Massy, FR;

Jean-Daniel Brion, Saint Leu la Foret, FR;

Jérôme Bignon, Le Val Saint Germain, FR;

Joëlle Dubois, Gometz-la-Ville, FR;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07C 69/734 (2006.01); C07C 235/64 (2006.01); C07D 209/42 (2006.01); C07D 213/65 (2006.01); A61K 45/06 (2006.01); C07D 239/74 (2006.01); C07C 235/38 (2006.01); C07D 215/14 (2006.01); C07C 259/06 (2006.01); C07D 213/81 (2006.01); C07C 259/10 (2006.01); C07D 209/86 (2006.01); A61K 47/68 (2017.01); A61P 35/00 (2006.01); A61K 31/165 (2006.01); A61K 31/166 (2006.01); A61K 31/167 (2006.01); A61K 31/192 (2006.01); A61K 31/216 (2006.01); A61K 31/404 (2006.01); A61K 31/44 (2006.01); C07C 59/68 (2006.01); C07C 235/34 (2006.01); C07C 235/60 (2006.01); C07D 209/18 (2006.01);
U.S. Cl.
CPC ...
C07C 69/734 (2013.01); A61K 31/165 (2013.01); A61K 31/166 (2013.01); A61K 31/167 (2013.01); A61K 31/192 (2013.01); A61K 31/216 (2013.01); A61K 31/404 (2013.01); A61K 31/44 (2013.01); A61K 45/06 (2013.01); A61K 47/6803 (2017.08); A61P 35/00 (2018.01); C07C 59/68 (2013.01); C07C 235/34 (2013.01); C07C 235/38 (2013.01); C07C 235/60 (2013.01); C07C 235/64 (2013.01); C07C 259/06 (2013.01); C07C 259/10 (2013.01); C07D 209/18 (2013.01); C07D 209/42 (2013.01); C07D 209/86 (2013.01); C07D 213/65 (2013.01); C07D 213/81 (2013.01); C07D 215/14 (2013.01); C07D 239/74 (2013.01);
Abstract

The present invention relates to the design of novel molecules, referred to as 'multi-target' molecules, having a double pharmacophore and acting both as inhibitors of histone deacetylases (HDACs) and as inhibitors of tubulin polymerisation. The invention also describes the method for synthesising the 'multi-target' molecules and their use in the treatment of cancer, a pharmaceutical composition comprising at least one “multi-target” molecule, and the use of such compositions in the treatment of cancer.


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