The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 02, 2021

Filed:

Sep. 12, 2017
Applicant:

The Regents of the University of California, Oakland, CA (US);

Inventors:

Alan M. Fogelman, Los Angeles, CA (US);

Srinivasa T. Reddy, Cerritos, CA (US);

Mohamad Navab, Los Angeles, CA (US);

Assignee:
Attorneys:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 38/04 (2006.01); A61K 9/14 (2006.01); A61K 9/16 (2006.01); C12N 15/82 (2006.01); A61K 9/00 (2006.01); A61K 38/17 (2006.01); C07K 14/775 (2006.01);
U.S. Cl.
CPC ...
A61K 38/04 (2013.01); A61K 9/0053 (2013.01); A61K 9/141 (2013.01); A61K 9/1635 (2013.01); A61K 38/1709 (2013.01); C07K 14/775 (2013.01); C12N 15/8241 (2013.01); C12N 15/8257 (2013.01); A61K 9/1617 (2013.01);
Abstract

In various embodiments, ezetimibe-associated apoA-I mimetic peptide are provided that show improved synergistic activity between ezetimibe and the apoA-I peptide in vivo. In certain embodiments the peptide component is a transgenic 6F and the ezetimibe-associated apoA-I mimetic peptide is an Ez-T6F peptide. Methods of making the Ez-apoA-I peptides are also provided. In certain embodiments the methods involve incubating ezetimibe and an apoAI mimetic peptide (e.g., T6F) in a solution comprising ethyl acetate and acetic acid or in a solution comprising ethyl lactate and lactic acid; and drying the solution to provide a dry ezetimibe-associated apoA-I mimetic peptide.


Find Patent Forward Citations

Loading…