The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 12, 2021

Filed:

Jul. 08, 2019
Applicant:

60 Degrees Pharmaceuticals Llc, Washington, DC (US);

Inventors:

Geoffrey S. Dow, Washington, DC (US);

Bryan L. Smith, Chevy Chase, MD (US);

John P. Jones, Richmond, VA (US);

Moshe Shmuklarsky, Bethesda, MD (US);

Budda Balasubrahmanyam, Richmond, VA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/4706 (2006.01); C07D 215/40 (2006.01); A61P 33/06 (2006.01);
U.S. Cl.
CPC ...
A61K 31/4706 (2013.01); A61P 33/06 (2018.01); C07D 215/40 (2013.01); Y02A 50/411 (2018.01);
Abstract

Methods of prevention of symptomatic malaria in a malaria-naïve, G6PD-normal human subject comprising administering to the human subject a compound of Formula (I), a pharmaceutically acceptable salt thereof, or pharmaceutical composition comprising a compound of Formula (I). A compound of Formula (I) can be administered prior to potential exposure of a species of, during potential exposure of a species of, and after potential exposure of a species of. The methods of the invention also pertains to kits comprising specific doses of Formula (I), a pharmaceutically acceptable salt thereof, or pharmaceutical composition comprising a compound of Formula (I), and instructions for administration of dosing quantity and frequency. The methods of the invention also pertain to determining doses of Formula (I) that meet the general regulatory requirement for a drug to be efficacious in the prevention of malaria in malaria-naïve subjects. The methods of the invention further pertain to using the described algorithm to derive dosing regimens which can provide protection against symptomatic malaria in malaria-naïve, G6PD-normal subjects.


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