The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Dec. 15, 2020
Filed:
Sep. 11, 2013
Merck Sharp & Dohme Corp., Rahway, NJ (US);
Lawrence Livermore National Security, Llc, Livermore, CA (US);
Daniel Bensen, Carlsbad, CA (US);
Allen Borchardt, San Diego, CA (US);
Zhiyong Chen, San Diego, CA (US);
John M. Finn, Encinitas, CA (US);
Thanh To Lam, San Diego, CA (US);
Suk Joong Lee, San Diego, CA (US);
Xiaoming Li, San Diego, CA (US);
Leslie William Tari, San Diego, CA (US);
Min Teng, San Diego, CA (US);
Michael Trzoss, San Diego, CA (US);
Junhu Zhang, San Diego, CA (US);
Michael E. Jung, Los Angeles, CA (US);
Felice C. Lightstone, Fremont, CA (US);
Sergio E. Wong, San Jose, CA (US);
Toan B. Nguyen, San Ramon, CA (US);
MERCK SHARP & DOHME CORP., Rahway, NJ (US);
LAWRENCE LIVERMORE NATIONAL SECURITY, LLC, Livermore, CA (US);
Abstract
Disclosed herein are compounds having the structure of Formula I and pharmaceutically suitable salts, esters, and prodrugs thereof that are useful as antibacterially effective tricyclic gyrase inhibitors. In addition, species of tricyclic gyrase inhibitors compounds are also disclosed herein. Related pharmaceutical compositions, uses and methods of making the compounds are also contemplated.