The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 24, 2020

Filed:

Feb. 13, 2020
Applicants:

The Johns Hopkins University, Baltimore, MD (US);

Lieber Institute, Inc., Baltimore, MD (US);

Inventors:

Pankaj Pasricha, Ellicott City, MD (US);

Yifang Huang, Lansdale, PA (US);

James Barrow, Arnold, MD (US);

Assignees:

The Johns Hopkins University, Baltimore, MD (US);

Lieber Institute, Inc., Baltimore, MD (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/5517 (2006.01); A61K 31/5513 (2006.01); A61K 45/06 (2006.01); A61P 25/00 (2006.01); C07D 243/12 (2006.01); C07D 243/24 (2006.01); C07D 487/04 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); A61K 31/5513 (2013.01); A61K 31/5517 (2013.01); A61K 45/06 (2013.01); C07D 243/12 (2013.01); C07D 243/24 (2013.01);
Abstract

The present invention provides compounds and compositions which are positive allosteric modulators of GABA-A receptors that selectively target the peripheral nervous system and organs of the body, and which do not pass through the blood-brain barrier. The compounds and compositions of the present invention are useful for treatment of diseases or disorders which are mediated by GABA-A neuronal activity, such as, for example, visceral pain, gut motility, irritable bowel syndrome, functional abdominal pain, functional idiopathic diarrhea, inflammatory bowel diseases, drug induced pain, bile salt malabsorption, lactase or other carbohydrate intolerance.


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