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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10807970 B1

PDFFull Text
Expired
Date of Patent:
Oct. 20, 2020

Filed:

May. 19, 2017

Tetrahydropyran and thiopyran derivatives having multimodal activity against pain

Applicant:

Esteve Pharmaceuticals, S.a., Barcelona, ES;

Inventors:

Monica Garcia-Lopez, Barcelona, ES;

Carmen Almansa-Rosales, Barcelona, ES;

Ana Virginia Llorente-Fernandez, Barcelona, ES;

Ute Christmann, Barcelona, ES;

Sergio Rodriguez Escrich, Barcelona, ES;

Assignee:

ESTEVE PHARMACEUTICALS, S.A., Barcelona, ES;

Attorney:

Hueschen and Sage

Primary Examiner:

Mark L Shibuya

Assistant Examiner:

Ebenezer O Sackey

Int. Cl.
CPC ...
C07D 405/04 (2006.01); C07D 405/14 (2006.01); C07D 487/04 (2006.01); A61P 29/00 (2006.01); C07D 307/04 (2006.01); C07D 407/14 (2006.01); C07D 407/06 (2006.01);
U.S. Cl.
CPC ...
C07D 405/04 (2013.01); A61P 29/00 (2018.01); C07D 307/04 (2013.01); C07D 405/14 (2013.01); C07D 407/06 (2013.01); C07D 407/14 (2013.01); C07D 487/04 (2013.01);
Abstract

The present invention relates to tetrahydropyran and thiopyran derivatives having dual pharmacological activity towards both the sigma (σ) receptor, and the μ-opioid receptor, to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy, in particular for the treatment of pain.

Find Patent Forward Citations

Garcia-Lopez, Monica. (2020). Tetrahydropyran and thiopyran derivatives having multimodal activity against pain (U.S. Patent No. 10807970). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/10807970

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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