The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 13, 2020

Filed:

Sep. 15, 2017
Applicant:

Entasis Therapeutics Limited, Altrincham, Cheshire, GB;

Inventors:

Janelle Comita-Prevoir, Northborough, MA (US);

Thomas Francois Durand-Reville, Belmont, MA (US);

Lise Gauthier, Waltham, MA (US);

John O'Donnell, Mattapoisett, MA (US);

Jan Romero, Arlington, MA (US);

Ruben Tommasi, Stow, MA (US);

Jeroen Cunera Verheijen, Westborough, MA (US);

Frank Wu, Shrewsbury, MA (US);

Xiaoyun Wu, Westborough, MA (US);

Jing Zhang, Sudbury, MA (US);

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 471/08 (2006.01); C07D 211/78 (2006.01); A61P 31/04 (2006.01); A61K 31/546 (2006.01); A61K 45/06 (2006.01); A61K 31/46 (2006.01); A61K 31/439 (2006.01);
U.S. Cl.
CPC ...
C07D 471/08 (2013.01); A61K 31/439 (2013.01); A61K 31/46 (2013.01); A61K 31/546 (2013.01); A61K 45/06 (2013.01); A61P 31/04 (2018.01); C07D 211/78 (2013.01); Y02A 50/404 (2018.01); Y02A 50/406 (2018.01); Y02A 50/473 (2018.01);
Abstract

The present invention is directed to compounds which are beta-lactamase inhibitors. The compounds and their pharmaceutically acceptable salts are useful in combination with beta-lactam antibiotics, for the treatment of bacterial infections, including infections caused by drug resistant organisms, including multi-drug resistant organisms. The present invention includes compounds according to Formula (I): or a pharmaceutically acceptable salt thereof, wherein the values of R, R, R, R, Rand Rare described herein.


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