The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 14, 2020

Filed:

Oct. 24, 2017
Applicant:

Hangzhou Hertz Pharmaceutical Co., Ltd., Hangzhou, Zhejiang Province, CN;

Inventors:

Xinglu Zhou, Hangzhou, CN;

Xingguo Liu, Hangzhou, CN;

Miao Hu, Hangzhou, CN;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/519 (2006.01); C07D 487/04 (2006.01); A61P 37/06 (2006.01); A61P 19/02 (2006.01); A61P 35/00 (2006.01); A61P 21/04 (2006.01); A61K 45/06 (2006.01); A61P 1/00 (2006.01); A61P 17/00 (2006.01); A61P 35/02 (2006.01); A61P 37/02 (2006.01); A61P 3/10 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); A61K 31/519 (2013.01); A61K 45/06 (2013.01); A61P 1/00 (2018.01); A61P 3/10 (2018.01); A61P 17/00 (2018.01); A61P 19/02 (2018.01); A61P 21/04 (2018.01); A61P 35/00 (2018.01); A61P 35/02 (2018.01); A61P 37/02 (2018.01); A61P 37/06 (2018.01);
Abstract

The present invention relates to a selective Bruton's tyrosine kinase (BTK) inhibitor compound, a pharmaceutical composition, preparation and use thereof in preparation of a drug. The compound of the present invention has a structure of Formula II or Formula II': Re is selected from H, CH, C2-C6 alkyl, C1-C6 azaalkyl, and C1-C6 oxaalkyl, wherein CH, C2-C6 alkyl, C1-C6 azaalkyl and C1-C6 oxaalkyl are further substituted with amino, hydroxyl, and C1-C3 alkyl;Y, Y, Yand Yare independently selected from C(Rf) and N, and at least one of Y, Y, Yand Yis N, wherein Rf is selected from H, halogen, C1-C3 alkyl, —CF, and —CFH.


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