The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 30, 2020

Filed:

Dec. 20, 2017
Applicant:

Research Triangle Institute, Research Triangle Park, NC (US);

Inventors:

Rangan Maitra, Cary, NC (US);

Robert W. Wiethe, Durham, NC (US);

Yanan Zhang, Apex, NC (US);

George S. Amato, Cary, NC (US);

Assignee:

Research Triangle Institute, Research Triangle Park, NC (US);

Attorneys:
Int. Cl.
CPC ...
C07D 473/34 (2006.01); C07D 471/10 (2006.01); A61K 31/52 (2006.01); A61P 1/16 (2006.01);
U.S. Cl.
CPC ...
C07D 473/34 (2013.01); A61K 31/52 (2013.01); A61P 1/16 (2018.01); C07D 471/10 (2013.01);
Abstract

This disclosure is directed to various compounds and methods of preparation of improved compounds that are capable of functioning as cannabinoid receptor 1 (CB1) antagonists with reduced central nervous system (CNS) side effects. The application is also directed to pharmaceutical compositions containing one or more of these compounds, which may also contain one or more additional therapeutic agents. It is also directed to methods of treatment of various conditions that may be responsive to antagonism of the CB1 receptors, including, but not limited to, metabolic syndromes (including liver disease, obesity, and diabetes).


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