The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 16, 2020

Filed:

Oct. 12, 2018
Applicant:

Jiangnan University, Wuxi, Jiangsu, CN;

Inventors:

Liping Zhang, Jiangsu, CN;

Caihua Ni, Jiangsu, CN;

Ren Liu, Jiangsu, CN;

He Liu, Jiangsu, CN;

Xinyi Dong, Jiangsu, CN;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 9/107 (2006.01); C08G 81/00 (2006.01); A61K 31/704 (2006.01); C08G 83/00 (2006.01); C08G 69/10 (2006.01); C08G 69/42 (2006.01);
U.S. Cl.
CPC ...
A61K 9/1075 (2013.01); A61K 31/704 (2013.01); C08G 69/10 (2013.01); C08G 69/42 (2013.01); C08G 81/00 (2013.01); C08G 83/003 (2013.01);
Abstract

Hybrid amphiphilic star copolymer nano micelles are prepared in the invention. Cage shaped octa(γ-aminopropyl) silsesquioxanes is selected as the inorganic part, and L-glutamic benzyl ester—five membered ring anhydride is ring-opening polymerized by the initiation of amino groups on the surface of cage shaped octa(γ-aminopropyl) silsesquioxanes, producing copolymers with cage shaped octa(γ-aminopropyl) silsesquioxanes as nucleus and poly (L-glutamic-benzyl ester) as arms. The copolymers reacts with monomethoxy poly (ethylene glycol) carboxylic acid by condensation. Finally, the benzyl groups in the side chains of poly (L-glutamic acid-benzyl ester) are converted into hydrazine groups by acylhydrazination to obtain hybrid amphiphilic star copolymer nano micelles. The micelles can load doxorubicin, they are safe to human body and have good application prospects.


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