The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 19, 2020

Filed:

Nov. 03, 2016
Applicants:

Dana-farber Cancer Institute, Inc., Boston, MA (US);

The Brigham and Women's Hospital, Inc., Boston, MA (US);

Inventors:

Alan D. D'Andrea, Winchester, MA (US);

Gregory D. Cuny, Houston, TX (US);

Ross L. Stein, Cambridge, MA (US);

Marcie Glicksman, Winchester, MA (US);

April Case, Watertown, MA (US);

Jun Xian, Sharon, MA (US);

David Wilson, Lawrence, KS (US);

Min Huang, Shanghai, CN;

Assignees:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 31/423 (2006.01); C07D 405/06 (2006.01); C07D 263/60 (2006.01); A61K 31/136 (2006.01); A61K 31/472 (2006.01); A61K 31/4725 (2006.01); A61K 45/06 (2006.01); C07C 225/30 (2006.01); C07D 217/24 (2006.01);
U.S. Cl.
CPC ...
A61K 31/423 (2013.01); A61K 31/136 (2013.01); A61K 31/472 (2013.01); A61K 31/4725 (2013.01); A61K 45/06 (2013.01); C07C 225/30 (2013.01); C07D 217/24 (2013.01); C07D 263/60 (2013.01); C07D 405/06 (2013.01);
Abstract

Provided are small molecule inhibitors of ubiquitin specific protease 1 (USP1) activity and methods for their use in treating and characterizing cancers. The small molecule USP1 inhibitors of the invention are particularly useful in the treatment of cancers that are resistant to DNA cross-linking agents.


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