The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 24, 2020

Filed:

Mar. 10, 2016
Applicant:

Shionogi Inc., Florham Park, NJ (US);

Inventors:

Zhengming Chen, Belle Mead, NJ (US);

Xiaoming Chen, Westfield, NJ (US);

Kevin Halloran, Somerset, NJ (US);

Assignee:

Shionogi, Inc., Florham Park, NJ (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/085 (2006.01); A61K 47/32 (2006.01); A61K 9/14 (2006.01); A61K 47/38 (2006.01);
U.S. Cl.
CPC ...
A61K 9/146 (2013.01); A61K 31/085 (2013.01); A61K 47/32 (2013.01); A61K 47/38 (2013.01);
Abstract

An ospemifene solid dispersion for enhancing solubility and bioavailability, and methods of preparation thereof are disclosed. The solid dispersion comprises an active pharmaceutical ingredient, such as ospemifene, and a hydfophilie carrier, such as copovidone, hypromellose acetate succinate, polyvinylpyrrolidine, a polyvinylpyrrolidine/vinyl acetate co-polymer, hydroxyl propyl methylcellulose, hypromellose acetate succinate, a Eudragit® compound, hydroxypropylcellulose, a polyvinyl caprolactam-polyvinyl acetate polyethylene glycol graft co-polymer, hydroxypropyl methylcellulose phthalate, and mixtures thereof, and optionally a surfactant The ospemifene solid, dispersions can be used in methods of treating a symptom related, to menopause, such as vaginal dryness or sexual dysfunction, or in methods of treating osteoporosis.


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