The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 17, 2020

Filed:

Jun. 29, 2016
Applicant:

William Marsh Rice University, Houston, TX (US);

Inventors:

Kyriacos C. Nicolaou, Houston, TX (US);

Ruofan Li, Houston, TX (US);

Zhaoyong Lu, Houston, TX (US);

Te-ik Sohn, Andong, KR;

James Woods, Houston, TX (US);

Emmanouil N. Pitsinos, Houston, TX (US);

Assignee:

WILLIAM MARSH RICE UNIVERSITY, Houston, TX (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07H 15/24 (2006.01); A61K 45/06 (2006.01); C07D 471/04 (2006.01); C07D 405/06 (2006.01); C07D 519/00 (2006.01); C07H 15/203 (2006.01); A61K 47/68 (2017.01); C07H 15/20 (2006.01); C07D 487/04 (2006.01); A61P 35/00 (2006.01); A61K 31/706 (2006.01); C07D 498/10 (2006.01);
U.S. Cl.
CPC ...
C07H 15/24 (2013.01); A61K 31/706 (2013.01); A61K 45/06 (2013.01); A61K 47/6803 (2017.08); A61K 47/6807 (2017.08); A61P 35/00 (2018.01); C07D 405/06 (2013.01); C07D 471/04 (2013.01); C07D 487/04 (2013.01); C07D 498/10 (2013.01); C07D 519/00 (2013.01); C07H 15/20 (2013.01); C07H 15/203 (2013.01);
Abstract

In one aspect, the present disclosure provides shishijimicin analogs of the formula: wherein the variables are as defined herein. In another aspect, the present disclosure also provides methods of preparing the compounds disclosed herein. In another aspect, the present disclosure also provides pharmaceutical compositions and methods of use of the compounds disclosed herein. Additionally, antibody drug conjugates of the compounds are also provided.


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