The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 28, 2020

Filed:

Feb. 29, 2016
Applicants:

SI Chuan University, Sichua, CN;

Lijuan Chen, Sichuan, CN;

Inventors:

Lijuan Chen, Sichuan, CN;

Yuquan Wei, Sichuan, CN;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 409/04 (2006.01); C07D 311/16 (2006.01); C07D 405/04 (2006.01); C07D 409/14 (2006.01); C07D 409/12 (2006.01); C07D 407/12 (2006.01); A61P 35/00 (2006.01);
U.S. Cl.
CPC ...
C07D 409/04 (2013.01); A61P 35/00 (2018.01); C07D 311/16 (2013.01); C07D 405/04 (2013.01); C07D 407/12 (2013.01); C07D 409/12 (2013.01); C07D 409/14 (2013.01);
Abstract

The present invention pertains to the field of chemical medicine, particularly to 4-substituted coumarin derivatives and preparation methods and applications thereof. The invention provides 4-substituted coumarin derivatives with a structural formula as shown in Formula I. The invention also provides preparation methods and applications for the above 4-substituted coumarin derivatives. The compounds provided in the invention have strong anti-tumor activity with IC50 for plural tumor cell lines between 0.01-5 nM, and it also performs better to inhibit microtubule polymerization and has diversified biological activities and low toxicity, providing new options for drug-sensitive and drug-resistant tumor cells.


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