The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 28, 2020

Filed:

Nov. 24, 2016
Applicant:

Hovione Scientia Limited, Cork, IE;

Inventors:

Luis Sobral, Loures, PT;

Livia Santana De Arruda, Rio de Janeiro, BR;

Margarida Figueiredo, Pinhal Novo, PT;

Rafael Antunes, Setubal, PT;

Ana Paula Filipe, Loures, PT;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61L 29/16 (2006.01); C07C 231/12 (2006.01); C07C 237/26 (2006.01); A61L 31/16 (2006.01); A61K 31/65 (2006.01);
U.S. Cl.
CPC ...
A61L 29/16 (2013.01); A61L 31/16 (2013.01); C07C 231/12 (2013.01); C07C 237/26 (2013.01); A61K 31/65 (2013.01); A61L 2300/406 (2013.01); A61L 2300/41 (2013.01);
Abstract

A tetracycline salt comprising a tetracycline and an organic acid wherein the organic acid is oxalic acid or maleic acid is provided. The tetracycline is preferably doxycycline, minocycline, sancycline, lymecycline, tetracycline or demeclocycline, and preferred salts include oxycycline maleate, minocycline oxalate, tetracycline oxalate, demeclocycline maleate, demeclocycline oxalate, sancycline maleate, lymecycline maleate, or lymecycline oxalate. A pharmaceutical formulation comprising a tetracycline salt according to the invention is also provided, as is a medical device having coated thereon a salt or pharmaceutical formulation according to the invention. A salt of the invention, or a formulation of the invention are also provided for use as medicaments, particularly for use in the treatment or prevention of an inflammation and/or an infection. There is also provided a method of preparing a tetracycline salt, which method comprises reacting a tetracycline base with an excess of an organic acid in a solvent.


Find Patent Forward Citations

Loading…