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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10532995 B1

PDFFull Text
Date of Patent:
Jan. 14, 2020

Filed:

Feb. 29, 2016

Substituted pyrazole compounds as serine protease inhibitors

Applicant:

Verseon Corporation, Fremont, CA (US);

Inventors:

Kevin Michael Short, Fremont, CA (US);

Maria de los Angeles Estiarte-Martinez, Fremont, CA (US);

David Ben Kita, Fremont, CA (US);

Timothy Philip Shiau, Fremont, CA (US);

Assignee:

VERSEON CORPORATION, Fremont, CA (US);

Attorney:

Davis Wright Tremaine LLP

Primary Examiner:

Taofiq A Solola

Int. Cl.
CPC ...
C07D 403/04 (2006.01); C07D 409/14 (2006.01); C07D 417/14 (2006.01); A61K 9/00 (2006.01); A61K 31/4155 (2006.01); A61K 31/454 (2006.01); A61K 31/4545 (2006.01); A61K 31/5377 (2006.01); A61K 31/55 (2006.01); A61K 45/06 (2006.01); C07D 401/04 (2006.01); C07D 405/04 (2006.01); C07D 405/14 (2006.01);
U.S. Cl.
CPC ...
C07D 403/04 (2013.01); A61K 9/0019 (2013.01); A61K 9/0048 (2013.01); A61K 31/4155 (2013.01); A61K 31/454 (2013.01); A61K 31/4545 (2013.01); A61K 31/5377 (2013.01); A61K 31/55 (2013.01); A61K 45/06 (2013.01); C07D 401/04 (2013.01); C07D 405/04 (2013.01); C07D 405/14 (2013.01); C07D 409/14 (2013.01); C07D 417/14 (2013.01);
Abstract

There are provided inter alia multisubstituted aromatic compounds useful for the inhibition of thrombin and/or kallikrein, which compounds include substituted pyrazolyl. There are additionally provided pharmaceutical compositions. There are additionally provided methods of treating and preventing certain diseases or disorders, which diseases or disorders are amenable to treatment or prevention by the inhibition of thrombin and/or kallikrein.

Find Patent Forward Citations

Short, Kevin. (2020). Substituted pyrazole compounds as serine protease inhibitors (U.S. Patent No. 10532995). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/10532995

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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