The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10494383 B1

PDF
Full Text
Expired
Date of Patent:
Dec. 03, 2019

Filed:

Jun. 23, 2017
Applicant:

Dalian University of Technology, Dalian, Liaoning, CN;

Inventors:

Yuhan Zhou, Liaoning, CN;

Jingping Qu, Liaoning, CN;

Yang Liu, Liaoning, CN;

Yilong Zhao, Liaoning, CN;

Assignee:

DALIAN UNIVERSITY OF TECHNOLOGY, Dalian, Liaoning, CN;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07C 45/40 (2006.01); C07C 45/68 (2006.01); C07C 69/74 (2006.01); C07F 5/00 (2006.01); C07F 5/02 (2006.01); C07C 69/76 (2006.01);
U.S. Cl.
CPC ...
C07F 5/02 (2013.01); C07C 45/40 (2013.01); C07C 45/68 (2013.01); C07C 69/76 (2013.01); C07F 5/025 (2013.01); C07C 2603/74 (2017.05);
Abstract

The present invention relates to a method for preparing difluoroallylboronate and application thereof, and it belongs to a field of compound preparation. A method for preparing difluoroallyl borate ester is using a compound of the formula II and bis (pinacolato) diboron as raw materials in a solvent and in the presence of an iron catalyst and a base according to the following reaction formula, to obtain a compound of the formula I, The method of the present invention directly use an inexpensive, commercially available metal iron salt as a catalyst to provide a convenient, low-cost method for preparing difluoroallyl borate ester, and provide a new and effective approach for the synthesis of γ-aminobutyric acid receptor agonist (III).


Find Patent Forward Citations

Zhou, Yuhan. (2019). Method for preparing difluoroallylboronate and application thereof (U.S. Patent No. 10494383). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/10494383

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