The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 10, 2019

Filed:

Sep. 01, 2016
Applicant:

Howard Hughes Medical Institute, Chevy Chase, MD (US);

Inventors:

Luke D. Lavis, Leesburg, VA (US);

Jonathan B. Grimm, Ashburn, VA (US);

Laurel M. Heckman, Ashburn, VA (US);

Eric R. Schreiter, Leesburg, VA (US);

Assignee:

HOWARD HUGHES MEDICAL INSTITUTE, Chevy Chase, MD (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 311/16 (2006.01); C07D 307/94 (2006.01); C07D 311/82 (2006.01); C07D 405/12 (2006.01); A61N 5/06 (2006.01); A61K 41/00 (2006.01); C09K 11/06 (2006.01); G01N 21/64 (2006.01); G01N 33/58 (2006.01); G01N 33/84 (2006.01);
U.S. Cl.
CPC ...
C07D 311/16 (2013.01); A61K 41/0057 (2013.01); A61N 5/06 (2013.01); A61N 5/062 (2013.01); C07D 307/94 (2013.01); C07D 311/82 (2013.01); C07D 405/12 (2013.01); C09K 11/06 (2013.01); G01N 21/6428 (2013.01); G01N 33/582 (2013.01); G01N 33/84 (2013.01); C09K 2211/1022 (2013.01); G01N 2021/6439 (2013.01);
Abstract

The presently-disclosed subject matter relates to analyte-activated photolabile compounds. The compounds include the formula: wherein Z includes a maskable molecule; L is selected from a bond, C, C(O), O, alkyl, (O)alkyl, and alkoxy; Ris selected from H, halogen, alkyl, and acyl; each Ris independently selected from H, alkyl, aryl, and acyl, and is optionally substituted with one or more heteroatoms independently selected from COOH and COO(alkyl); and Ris selected from H, alkyl, aryl, halogen, CN, OH, O(alkyl), O(aryl), SH, S(alkyl), S(aryl), amine, CHO, COOH, COO(alkyl), COO(aryl), POH, and SOH, and is optionally substituted with one or more heteroatoms independently selected from N, O, and S, halogen, OH, O(alkyl), O(aryl), SH, S(alkyl), S(aryl), amine, NO, CHO, COO, COOH, COO(alkyl), COO(aryl), C(O)NR, POH, and/or SOH. Also provided are methods of detecting calcium and treating a subject with the analyte-activated photolabile compounds.


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