The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Aug. 13, 2019

Filed:

Apr. 27, 2016
Applicant:

Jina Pharmaceuticals, Inc., Libertyville, IL (US);

Inventors:

Ateeq Ahmad, Wadsworth, IL (US);

Shoukath M. Ali, Vernon Hills, IL (US);

Moghis U. Ahmad, Wadsworth, IL (US);

Saifuddin Sheikh, Waukegan, IL (US);

Imran Ahmad, Libertyville, IL (US);

Assignee:

Jina Pharmaceuticals, Inc., Libertyville, IL (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 9/20 (2006.01); A61K 9/48 (2006.01); A61K 31/138 (2006.01); A61K 9/19 (2006.01); A61K 9/127 (2006.01); A61K 9/00 (2006.01); A61K 31/35 (2006.01); C07D 309/10 (2006.01);
U.S. Cl.
CPC ...
A61K 31/138 (2013.01); A61K 9/0014 (2013.01); A61K 9/127 (2013.01); A61K 9/19 (2013.01); A61K 9/20 (2013.01); A61K 9/48 (2013.01); A61K 31/35 (2013.01); C07D 309/10 (2013.01);
Abstract

The present invention provides compositions containing endoxifen, formulations and liposomes of endoxifen, methods of preparation of such agents and formulations, and use of such agents and formulations for the treatment of breast cancer and other breast diseases and diseases susceptible to endoxifen. In particular, the compositions of the present invention include liposomes, complexes, vesicles, emulsions, micelles and mixed micelles of endoxifen in which the compositions further contain any of a variety of neutral or charged lipids and desirably, cholesterol and cholesterol derivatives, sterols, Z- and E-guggulsterones, phospholipids, fatty acids, vitamin D, and vitamin E. The present invention also provides methods of preparing endoxifen. The present invention provides methods for treating and preventing breast cancer and other breast related diseases by administrating novel formulations or compositions comprising a therapeutically effective amount of endoxifen.


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