The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 05, 2019

Filed:

Mar. 09, 2012
Applicants:

Hiroaki Suga, Tokyo, JP;

Yuki Goto, Tokyo, JP;

Yumi Ito, Tokyo, JP;

Inventors:

Hiroaki Suga, Tokyo, JP;

Yuki Goto, Tokyo, JP;

Yumi Ito, Tokyo, JP;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C12N 15/10 (2006.01); G01N 33/543 (2006.01); C12Q 1/37 (2006.01); C07K 14/47 (2006.01); C12P 21/02 (2006.01); C12P 17/16 (2006.01);
U.S. Cl.
CPC ...
G01N 33/54393 (2013.01); C07K 14/47 (2013.01); C12N 15/1062 (2013.01); C12P 21/02 (2013.01); C12Q 1/37 (2013.01); C12P 17/16 (2013.01); G01N 2500/00 (2013.01);
Abstract

An object of the present invention is to provide a method of efficiently constructing a library abundant in diversity and also usable for screening of a compound that binds to a target substance having protease activity. The present invention provides a method of constructing an azoline compound library containing two or more azoline compounds having an azoline backbone introduced into at least one of Cys, Ser, Thr, and 2,3-diamino acid, and analogs thereof of Xaaof a peptide represented by the following formula (I):A-(Xaa)-B  (I)[wherein, m numbers of Xaas respectively represent arbitrary amino acids, at least one of which is an amino acid selected from the group consisting of Cys, Ser, Thr, and 2,3-diamino acid, and analogs thereof, m represents an inter selected from 2 to 40, and A and B each independently represent a peptide composed of from 0 to 100 amino acids].


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