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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10138229 B1

PDFFull Text
Date of Patent:
Nov. 27, 2018

Filed:

Nov. 16, 2017

Heteroaromatic compounds as btk inhibitors

Applicant:

Boehringer Ingelheim International Gmbh, Ingelheim am Rhein, DE;

Inventors:

Joerg Bentzien, White Plains, NY (US);

Angela Kay Berry, Gaylordsville, CT (US);

Todd Bosanac, New Milford, CT (US);

Michael Jason Burke, Newtown, CT (US);

Darren Todd Disalvo, New Milford, CT (US);

Joshua Courtney Horan, Somerville, MA (US);

Shuang Liang, Roseville, MN (US);

Can Mao, Philadelphia, PA (US);

Wang Mao, Milford, CT (US);

Yue Shen, Ridgefield, CT (US);

Fariba Soleymanzadeh, Danbury, CT (US);

Renee M. Zindell, New Milford, CT (US);

Assignee:

Boehringer Ingelheim International GmbH, Ingelheim am Rhein, DE;

Attorney:

Atabak R. Royaee

Primary Examiner:

Kamal Saeed

Int. Cl.
CPC ...
C07D 403/04 (2006.01); C07D 403/06 (2006.01); C07D 403/08 (2006.01); C07D 231/14 (2006.01); C07D 413/14 (2006.01); C07D 401/04 (2006.01); C07D 401/14 (2006.01); C07D 401/02 (2006.01); C07D 277/56 (2006.01); C07D 231/40 (2006.01); C07D 231/38 (2006.01); C07D 417/04 (2006.01); C07D 417/06 (2006.01); C07D 417/08 (2006.01); C07D 405/14 (2006.01); C07D 401/06 (2006.01); C07D 417/02 (2006.01);
U.S. Cl.
CPC ...
C07D 417/08 (2013.01); C07D 231/14 (2013.01); C07D 231/38 (2013.01); C07D 231/40 (2013.01); C07D 277/56 (2013.01); C07D 401/02 (2013.01); C07D 401/04 (2013.01); C07D 401/06 (2013.01); C07D 401/14 (2013.01); C07D 403/04 (2013.01); C07D 403/06 (2013.01); C07D 403/08 (2013.01); C07D 405/14 (2013.01); C07D 413/14 (2013.01); C07D 417/02 (2013.01); C07D 417/04 (2013.01); C07D 417/06 (2013.01);
Abstract

The present invention encompasses compounds of the formula (I) wherein the groups A, Cy, X1 and Y are defined herein, which are suitable for the treatment of diseases related to BTK, process of making, pharmaceutical preparations which contain compounds and their methods of use.

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