The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 13, 2018

Filed:

Aug. 25, 2016
Applicants:

The United States of America, As Represented BY the Secretary, Department of Health and Human Service, Washington, DC (US);

The Florida International University Board of Trustees, Miami, FL (US);

Inventors:

Juan Jose Marugan, Gaithersburgh, MD (US);

Jingbo Xiao, Rockville, MD (US);

Marc Ferrer-Alegre, Potomac, MD (US);

Catherine Chen, Germantown, MD (US);

Noel Southall, Potomac, MD (US);

Wei Zheng, Potomac, MD (US);

Alexander Agoulnik, Miami, FL (US);

Irina Agoulnik, Miami, FL (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 233/64 (2006.01); A61K 31/166 (2006.01); C07D 333/38 (2006.01); C07C 237/42 (2006.01); C07D 307/52 (2006.01); C07D 333/20 (2006.01); C07D 317/68 (2006.01); C07D 213/81 (2006.01); C07D 307/68 (2006.01); C07D 213/82 (2006.01); C07D 261/18 (2006.01); C07D 209/08 (2006.01); C07D 317/66 (2006.01); C07C 317/40 (2006.01); C07C 323/42 (2006.01); C07D 211/26 (2006.01); C07D 295/088 (2006.01); C07D 235/08 (2006.01); C07D 295/205 (2006.01); C07D 235/14 (2006.01); C07C 255/60 (2006.01); C07D 257/04 (2006.01); C07C 251/24 (2006.01);
U.S. Cl.
CPC ...
C07D 333/38 (2013.01); C07C 237/42 (2013.01); C07C 251/24 (2013.01); C07C 255/60 (2013.01); C07C 317/40 (2013.01); C07C 323/42 (2013.01); C07D 209/08 (2013.01); C07D 211/26 (2013.01); C07D 213/81 (2013.01); C07D 213/82 (2013.01); C07D 235/08 (2013.01); C07D 235/14 (2013.01); C07D 257/04 (2013.01); C07D 261/18 (2013.01); C07D 295/088 (2013.01); C07D 295/205 (2013.01); C07D 307/52 (2013.01); C07D 307/68 (2013.01); C07D 317/66 (2013.01); C07D 317/68 (2013.01); C07D 333/20 (2013.01);
Abstract

Disclosed are modulators of the human relaxin receptor 1, for example, of formula (I), wherein A, R, and Rare as defined herein, that are useful in treating mammalian relaxin receptor 1 mediated facets of human health, e.g., cardiovascular disease. Also disclosed is a composition comprising a pharmaceutically suitable carrier and at least one compound of the disclosure, and a method for therapeutic intervention in a facet of mammalian health that is mediated by a human relaxin receptor 1.


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