The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Aug. 14, 2018

Filed:

Aug. 25, 2015
Applicant:

Nippon Soda Co., Ltd., Chiyoda-ku, Tokyo, JP;

Inventor:

Shinichi Kobayashi, Takaoka, JP;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 223/06 (2006.01); C07C 221/00 (2006.01); C07D 317/16 (2006.01); C07D 317/28 (2006.01);
U.S. Cl.
CPC ...
C07C 223/06 (2013.01); C07C 221/00 (2013.01); C07D 317/16 (2013.01); C07D 317/28 (2013.01);
Abstract

The present invention provides a method for producing a benzaldehyde in which an amino group is bonded in the 2 position, a halogeno group or an alkoxy group is bonded in the 3 position, and a hydrogen atom, an alkyl group, a halogeno group, an alkoxy group, or a cyano group is bonded independently in each of the 4, 5, and 6 positions, the method including: preparing a benzaldehyde in which a halogeno group or an alkoxy group is bonded in the 3 position, a hydrogen atom is bonded in the 2 position, and a hydrogen atom, an alkyl group, a halogeno group, an alkoxy group, or a cyano group is bonded independently in each of the 4, 5, and 6 positions so that a lithiation reaction is most active at the 2 position; acetal-protecting a formyl group in the benzaldehyde; sequentially performing lithiation, azidation, and amination of the 2 position; and the performing acetal deportection.


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