The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 31, 2018

Filed:

Sep. 08, 2017
Applicant:

Jenkem Technology Co., Ltd. (Tianjin), Tianjin, CN;

Inventors:

Lihua Xu, Beijing, CN;

Xuan Zhao, Beijing, CN;

Zewang Feng, Beijing, CN;

Jinliang Wang, Beijing, CN;

Zhen'guo Wang, Beijing, CN;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 47/60 (2017.01); A61K 31/4045 (2006.01); A61K 31/506 (2006.01); A61K 31/00 (2006.01); A61K 31/382 (2006.01);
U.S. Cl.
CPC ...
A61K 47/60 (2017.08); A61K 31/00 (2013.01); A61K 31/382 (2013.01); A61K 31/4045 (2013.01); A61K 31/506 (2013.01);
Abstract

Provided are polyethylene glycol drug conjugates of general formula (I), (II) or (III) and pharmaceutical compositions and a use thereof. The conjugates are formed by combining low molecular weight polyethylene glycol with 2-4 drug molecules. The conjugates can interact with receptor dimers or polymers, thereby improving the in vivo distribution of the drug, changing the oil and water distribution coefficient, enhancing the pharmacological activity, reducing the blood-brain barrier permeability of the drug, and improving the bioavailability of the drug.


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