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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10004740 B1

PDFFull Text
Date of Patent:
Jun. 26, 2018

Filed:

Mar. 27, 2015

Prodrugs of hiv reverse transcriptase inhibitors

Applicant:

Merck Sharp & Dohme Corp., Rahway, NJ (US);

Inventors:

Christopher S. Burgey, Ambler, PA (US);

Jeffrey F. Fritzen, Pottstown, PA (US);

Jaume Balsells, North Wales, PA (US);

Mehul Patel, Blue Bell, PA (US);

Assignee:

Merck Sharp & Dohme Corp., Rahway, NJ (US);

Attorneys:

Carol S. Quagliato

John C. Todaro

Primary Examiner:

Venkataraman Balasubramanian

Int. Cl.
CPC ...
C07D 403/06 (2006.01); C07D 237/22 (2006.01); C07D 239/47 (2006.01); A61K 31/501 (2006.01); A61K 31/506 (2006.01); A61K 31/513 (2006.01); A61P 31/18 (2006.01); A61K 45/06 (2006.01);
U.S. Cl.
CPC ...
A61K 31/506 (2013.01); A61K 31/501 (2013.01); A61K 31/513 (2013.01); A61K 45/06 (2013.01); C07D 237/22 (2013.01); C07D 239/47 (2013.01); C07D 403/06 (2013.01);
Abstract

Compounds of Formula I are described: wherein Rand Rare defined herein. The compounds of Formula I are useful in the inhibition of HIV reverse transcriptase, the prophylaxis and treatment of infection by HIV, and the prophylaxis, delay in the onset or progression, and treatment of AIDS. The compounds can be employed as ingredients in pharmaceutical compositions, optionally in combination with other antivirals, immunomodulators, antibiotics or vaccines.

Find Patent Forward Citations

Burgey, Christopher. (2018). Prodrugs of hiv reverse transcriptase inhibitors (U.S. Patent No. 10004740). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/10004740

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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