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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 10000502 B1

PDFFull Text
Date of Patent:
Jun. 19, 2018

Filed:

Jan. 11, 2017

Substituted thiohydantoin derivatives as androgen receptor antagonists

Applicant:

Janssen Pharmaceutica NV, Beerse, BE;

Inventors:

Gilles Bignan, Bridgewater, NJ (US);

Peter J Connolly, New Providence, NJ (US);

Ian Hickson, Tyne & Wear, GB;

Lieven Meerpoel, Beerse, BE;

Vineet Pande, Vosselaar, BE;

Zhuming Zhang, Hillsborough, NJ (US);

Jonathan Branch, Hatfield, PA (US);

Christian Rocaboy, Murcia, ES;

Luis B Trabalón Escolar, Murcia, ES;

Assignee:

Janssen Pharmaceutica NV, Beerse, BE;

Attorney:

Baker & Hostetler LLP

Primary Examiner:

Shawquia Jackson

Int. Cl.
CPC ...
C07D 491/107 (2006.01); C07D 401/14 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01); C07D 401/04 (2006.01); C07D 409/14 (2006.01); C07D 451/02 (2006.01); C07D 451/06 (2006.01); C07D 487/04 (2006.01); C07D 491/044 (2006.01); C07D 491/048 (2006.01); A61K 9/00 (2006.01); A61K 31/4439 (2006.01); A61K 31/4545 (2006.01); A61K 31/46 (2006.01); A61K 31/506 (2006.01); A61K 31/5377 (2006.01); A61K 31/55 (2006.01); A61K 31/573 (2006.01); A61K 31/58 (2006.01);
U.S. Cl.
CPC ...
C07D 491/107 (2013.01); A61K 9/0053 (2013.01); A61K 31/4439 (2013.01); A61K 31/4545 (2013.01); A61K 31/46 (2013.01); A61K 31/506 (2013.01); A61K 31/5377 (2013.01); A61K 31/55 (2013.01); A61K 31/573 (2013.01); A61K 31/58 (2013.01); C07D 401/04 (2013.01); C07D 401/14 (2013.01); C07D 405/14 (2013.01); C07D 409/14 (2013.01); C07D 413/14 (2013.01); C07D 451/02 (2013.01); C07D 451/06 (2013.01); C07D 487/04 (2013.01); C07D 491/044 (2013.01); C07D 491/048 (2013.01);
Abstract

Disclosed are compounds, compositions and methods for treating of disorders that are affected by the antagonism of one or more androgen receptor types. Such compounds are represented by Formula (I) as follows: wherein Rand G are defined herein.

Find Patent Forward Citations

Quick Actions:

Bignan, Gilles. (2018). Substituted thiohydantoin derivatives as androgen receptor antagonists (U.S. Patent No. 10000502). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/10000502

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