Nihon Nohyaku Co., Ltd.

Bayer Cropscience Gmbh

Shinsuke Fujioka

Takashi Furuya

Masanori Tohnishi

Hayami Nakao

Akira Seo

Toshiaki Shimizu

Kazuyuki Sakata

Hideo Kanno

Eiji Kohno

Tateki Nishida

Akiyuki Suwa

Masayuki Morimoto

Minoru Yamaguchi

Kozo Machiya

Hiroto Harayama

Makoto Goto

Kenji Tsubata

Tsuyoshi Takemoto

Masahiro Uehara

Masayuki Kimura

Yoshihiro Matsuzaki

Noriaki Yasokawa

The substituted pyrazolecarboxanilide derivatives represented by of the formula (I) wherein Ris H, alkyl, alkylcarbonyl, alkenylcarbonyl, cycloalkyl, phenylalkyl, phenylcarbonyl and the like; Ris H, halogen, alkyl, CN, OH, alkoxy, phenoxy, phenylthio, phenylsulfonyl and the like; G is alkyl, alkenyl, alkynyl, cycloalkyl, C-Ccycloalkenyl and the like; Z is O or S; X is H, halogen, CN, NO, alkyl and the like; Yis H, alkyl, alkenyl, phenyl, alkoxyalkyl and the like; Yis H, halogen, CN, NO, OH, mercapto, amino, carboxyl, C-Calkyl, phenyl, phenoxy, heterocycle and the like, m is 1 or 2; and n is 1-3, and salts thereof exhibit a superior effect as agrohorticultural insecticides or acaricides.

Substituted pyrazolecarboxylic acid anilide derivative or salt thereof, intermediate thereof, agent for agricultural and horticultural use, and use thereof

Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein Ris H, Calkyl, halo Calkyl, or the like; Ris halogeno, Calkyl, or the like; G is Calkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

Substituted pyrazinecarboxylic acid anilide derivatives or salts thereof, intermediates of the same, pesticides for agricultural and horticultural use, and usage thereof

Disclosed is a phthalamide derivative represented by the general formula (I) or a salt thereof, which shows an excellent controlling effect for use as an agricultural or horticultural insecticide alone or in combination with other agricultural or horticultural insecticide, acaricide, nematicide, fungicide, herbicide, plant growth regulator, biopesticide or the like. 

Phthalamide derivative, agricultural or horticultural pesticide, and use of the pesticide

The present invention provides a substituted anilide derivative of formula (I): {wherein Z is a group of formula (II) or (III) (in these formulas, A is C-Calkylene, C-Calkenylene, etc., Ris H, halogen, &#x2014;C(R)&#x2550;NOR, (substituted) phenyl, (substituted) heterocyclic ring, -A-R, etc.; Ris H, C-Calkyl, etc.), Ris H, C-Calkyl, etc.; Ris H, F, fluoro C-Calkyl; Rf is F, fluoro C-Calkyl; 1 is 0 to 2; Y is halogen, (substituted) phenyl, (substituted) phenoxy, etc.; and m is 0 to 3}, an intermediate thereof, an agrohorticultural agent, and a method for the use thereof. The compound of the present invention exhibits, at a low dosage, high uptake and translocation from the root and an excellent insecticidal effect especially when applied to soil.

Substituted aromatic amide derivative, intermediate thereof, agrohorticultural insecticide containing thereof and method for the use thereof

The present invention relates to a substituted anilide derivative represented by general formula (I): 

Substituted N-phenyl-phenoxy nicotinic acid-(thio)amides and their use as herbicides

The present invention relates to an aromatic diamide derivative represented by the general formula (I): 

Aromatic diamide derivatives, chemicals for agricultural or horticultural use and usage thereof

Sulfonamide derivatives represented by general formula (I) or salts thereof; insecticides for agricultural and horticultural use containing the same as the active ingredient; and usage thereof: [wherein A is optionally substituted (C&#x2013;C)alkylene, (C&#x2013;C)alkenylene or the like; Ris H, optionally substituted (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl, (C&#x2013;C)cycloalkyl or the like; R, Rand Rare each H, (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl or the like, or Rand A or Rand Rmay form a 3- to 8-membered ring which may be interrupted by one to three atoms selected from among O, S and N; Q is C or N; X and Y are each halogen, CN, NO, (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl or the like; m is 0 to 2; n is 0 to 3; and two adjacent Xs or Ys on the aromatic ring may be united to form a fused ring]. The compounds exhibit excellent insecticidal activity against insect pests resistant to existing pesticides even when applied in dosages lower than those of similar pesticides.

Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof

The present invention relates to a phthalamide derivative represented by the general formula (I): wherein R, R, R, X, Y, m, and n are as defined in the disclosure, which can be used as the active ingredient in an agricultural or horticultural insecticide that exhibits an excellent insecticidal effect even when used in a small active-ingredient amount.

Phthalamide derivative, agricultural or horticultural insecticide, and method of use thereof

Aromatic diamide derivative represented by the general formula (I) or a salt thereof and agricultural/herticultural composition containing the same as the active ingredient,wherein Arepresents alkylene, alkenylene or alkynylene; B represents, CO&#x2014; or &#x2014;C(&#x2550;N&#x2014;OR)&#x2014; (wherein Rrepresents H, etc.); Rto Rrepresent each H, etc.; Qto Qrepresent each N or carbon; Y represents halogeno, etc.; m is from 0 to 5; and Zand Zrepresent each O or S.

Aromatic diamide derivatives or salts thereof, agricultural/horticultural chemicals and method of using the same

Phthalamide derivatives, or salt thereof agrohorticultural insecticide, and method for using the same

Phthalic acid diamide derivatives, fluorine-containing aniline compounds as starting material, agricultural and horticultural insecticides, and a method for application of the insecticides

Phthalic acid diamide derivatives fluorine-containing aniline compounds as starting material, agricultural and horticultural insecticides, and a method for application of the insecticides

There are disclosed a compound represented by the general formula (I): ##STR1## (wherein R, R.sup.1, X, Y and n are as defined in the specification), a pest controller containing said compound as an active ingredient, a pest control method using said controller, and an intermediate for producing the compound of the above general formula (I).

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Kawachinagano, Japan

Shinsuke Fujioka