Lexicon Pharmaceuticals, Inc.

Lexicon Pharmaceutical Inc.

Qiuling Song

Haiming Zhang

Wenxue Wu

Jie Yan

Shinya Iimura

Ross Mabon

Matthew Mangzhu Zhao

Bryce Alden Harrison

Ramanaiah C Kanamarlapudi

Nicole Cathleen Goodwin

Hugh Alfred Burgoon, Jr

Mark S Bednarz

Hugh Alfred Burgoon

Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.

Methods of preparing 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds

Methods of synthesizing sodium glucose co-transporter 2 inhibitors, as well as compounds useful therein, are disclosed. Particular inhibitors are compounds of formula I. 

Methods and compounds useful for the preparation of sodium glucose co-transporter 2 inhibitors

Methods of synthesizing sodium glucose co-transporter 2 inhibitors, as well as compounds useful therein, are disclosed. Particular inhibitors are compounds of formula I: 

1-phenyl-1H-pyrazole-based compounds

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Newark, DE, United States of America

Qiuling Song