Dow Agrosciences LLC

Corteva Agriscience LLC

University of Pittsburgh

Sanofi

Adama Makhteshim, Ltd.

Sanofi-Aventis

Vps-3, Inc.

Adama Makteshim Ltd.

Viamet Pharmaceuticals, Inc.

Nakyen Choy

Gregory T Whiteker

Daniel Knueppel

Ronald Ross, Jr

Fangzheng Li

Ricky Hunter

Gary D Crouse

Tony K Trullinger

David Anthony Demeter

Timothy P Martin

Joseph D Eckelbarger

Zoltan Laszlo Benko

Maurice C Yap

John F Daeuble, Sr

Erich W Baum

Ronald J Heemstra

Frank J Wessels

Michelle Bowerman Riener

Peter Vednor

Yuanming Zhu

Kaitlyn C Gray

Thomas Clarence Sparks

Monica Britt Olson

Jeffrey S Nissen

James M Renga

Kyle A DeKorver

Peter S Borromeo

Kyle A Dekorver

Patrick S Hanley

Nicholas R Babij

Adam W Sledeski

William Joel Hoekstra

Gary A Roth

Carl Vincent DeAmicis

Dennis Patrick Curran

Michael Thomas Sullenberger

Matthias Stefan Ober

Gary David Gustafson

Billy W Day

Yong Mi Choi-Sledeski

Gregory Bernard Poli

John F Daeuble

Thomas L Siddall

Erich J Molitor

Carl DeAMICIS

Kenneth E Stockman

Jeff Nissen

John J Shay, Jr

Jim M Renga

Raghavan Balachandran

Youseung Shin

Tina Staton

Tiffany Turner

Tom Sparks

Volker Derdau

Nicole Hough

Grant Von Wald

Charitha Madiraju

Patrick Wai-Kwok Shum

Harpal S Gill

Andrea Hillegass

Daniel I Knueppel

John J Shay

Kaitlyn Gary

Peter Borromeo

Jim Renga

Zoltan L Venko

Kyla A Dekorver

Ronald Ross

Michelle Riener

Jeffrey Nissen

Zoltan L Benko

David A Demeter

Kaitlyn Gray

Greg Whiteker

Monica B Olson

Carl Deamicis

Timothy Allen Ayers

This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Arthropoda, Mollusca, and Nematoda, processes to produce such molecules, intermediates used in such processes, pesticidal compositions containing such molecules, and processes of using such pesticidal compositions against such pests. These pesticidal compositions may be used, for example, as acaricides, insecticides, miticides, molluscicides, and nematicides. This document discloses molecules having the following formula (“Formula One”).

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Arthropoda, Mollusca, and Nematoda, processes to produce such molecules, intermediates used in such processes, pesticidal compositions containing such molecules, and processes of using such pesticidal compositions against such pests. These pesticidal compositions may be used, for example, as acaricides, insecticides, miticides, molluscicides, and nematicides. This document discloses molecules having the following formula ('Formula One'). 

Provided herein are 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation which may include the use of an alkali carbonate and an alkylating agent 

5-fluoro-4-imino-3(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation

4-Alkoxy-3-hydroxypicolinic acids may be conveniently prepared from 4,6-dibromo-3-hydroxypicolinonitrile in a series of chemical steps selected from bromo substitution, nitrile hydrolysis and halogen reduction that are conducted as a single pot process. 4,6-Dibromo-3-hydroxypicolinonitrile may be prepared from furfural in a series of chemical steps selected from cyano-amination, amine salt formation and bromination-rearrangement.

Processes for the preparation of 4-alkoxy-3-hydroxypicolinic acids

A fungicidal 4-methoxy-3-acetyloxypicolinamide may be conveniently prepared in processes that include the coupling together of 4-methoxy-3-acetyloxypicolinic acid or 4-methoxy-3-hydroxypicolinic acid with a key 2-aminopropanoate ester derived from a 1,1-bis(4-fluorophenyl)propane-1,2-diol.

Processes for the preparation of 4-alkoxy-3-(acyl or alkyl)oxypicolinamdes

Provided herein are 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ols and 1-(2,4-difluorophenyl)-2,2-difluoro-2-(5-substituted-pyridin-2-yl)ethanones and processes for their preparation.

2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1h-tetrazol-1-yl)propan-2-ols and processes for their preparation

The (1R,3R)- or (1S,3S)-enantiomer of 2,2-dichloro-3-(substituted phenyl)cyclopropane-carboxylic acid is prepared in a process involving chemical resolution of a racemic mixture of a trans-2,2-dichloro-3-(substituted phenyl)cyclopropanecarboxylic acid with an enantiomeric amine, isolation of a diastereomeric amine salt and finally treatment of the salt with an acid.

Process for the preparation of (1R,3R)- and (1S,3S)-2,2-dihalo-3-(substituted phenyl)cyclopropanecarboxylic acids

Processes for the preparation of 4-alkoxy-3-(acyl or alkyl)oxypicolinamides

2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ols and processes for their preparation

4-Alkoxy-3-hydroxypicolinic acids may be conveniently prepared from 2-hydroxypicolinonitrile in a series of chemical steps selected from chlorination, chloro substitution, nitrile hydrolysis and chloro reduction.

Process for the preparation of 4-alkoxy-3-hydroxypicolinic acids

5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1 H)-one and processes for their preparation

Provided herein are 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)3,4-dihydropyrimidin-2(1H)-one and processes for their preparation which may include the use of an alkali alkoxide and an alkylating agent 

5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation

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Carmel, IN, United States of America

Nakyen Choy