Basf Se Corporation

Basf Agro B.v. Arnhem (nl), Zurich Branch

Maximilian Dochnahl

Michael Rack

Bernd Wolf

Timo Frassetto

Joachim Gebhardt

Uwe Josef Vogelbacher

Volker Maywald

Michael Keil

Roland Goetz

Frederik Menges

Roland Götz

Bernd Mueller

Karsten Koerber

Bernd Müller

Gunter Lipowsky

Jens Renner

Florian Kaiser

Prashant Deshmukh

Karsten Körber

Martin Sukopp

Alexander Korte

Philip Muelheims

Gemma Veitch

Rudolf Haeberle

Roland Gotz

Philip MÜLHEIMS

Rudolf HÄBERLE

Roland GÖTZ

The present invention relates to a process for preparing an N-substituted 1H-pyrazole-5-carboxylate compound of the formula (I-A) comprising the steps of  

Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof

The present invention relates to a process for manufacturing haloacetamides of formula (I), comprising

Process for manufacturing haloacetamides

The present invention relates to a process for manufacturing benzoxazinones of formula (I), wherein the variables are defined according to the description,by reacting carbamates of formula (II) are reacted with carbamat-benzoxazinones of formula (III) in the presence of a base.

Process for manufacturing benzoxazinones

The present invention relates to a process for manufacturing 4-propargylated amino-benzoxazinones of formula (I), comprising the following steps:

Process for manufacturing 4-propargylated amino-benzoxazinones

The present invention relates to carbamates of formula (I), 

Carbamates

The present invention relates to a process for manufacturing aryloxyacetamides of formula (I), by reacting haloacetamides of formula (II) with a phenol of formula (III); wherein the variables are defined according to the description, and aryloxyacetamides of formula (I).

Process for manufacturing aryloxyacetamides

The present invention relates to a process for manufacturing a benzoxazinone of formula (I), by reacting a nitro compound of formula (II) with a reducing agent to obtain an amino compound of formula (III), and then reacting the amino compound of formula (III) with an acid; wherein the variables are defined according to the description, and benzoxazinone of formula (I).

The present invention relates to carbamat-benzoxazinones of formula (I), wherein the variables are defined according to the description,

Carbamat-benzoxazinones

The present invention relates to a process using Grignard reagents for providing thio-triazolo group-containing compounds.

Process using Grignard reagents

The present invention relates to a process for manufacturing fluoroaromatics of formula (I),A-F &#x2003;&#x2003;(I)comprising

Process for manufacturing fluoroaromatics

The present invention relates to a process for manufacturing 4-substituted amino-benzoxazinones of formula (I), by reacting a NH-benzoxazinone of formula (II) with a compound of formula (III); wherein the variables are defined according to the description.

Process for manufacturing 4-substituted amino-benzoxazinones

The present invention relates to a process for manufacturing triazinon-benzoxazinones of formula (I), by reacting amino-benzoxazinones of formula (II) with 1,1'-carbonyldiimidazole (CDI) and a (thio)urea compound of formula (III); wherein the variables are defined according to the description.

Process for manufacturing triazinon-benzoxazinones

The present invention to a process for preparing 1-phenylpyrazoles of the formula I in which each Ris independently selected from chlorine, fluorine, alkyl, haloalkyl, alkoxy and haloalkoxy; n is 1, 2 or 3; each Ris independently selected from cyano, nitro, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio and alkoxycarbonyl; m is 0, 1 or 2; A is alkyl, aryl or aryl-C-C-alkyl, where A optionally bears 1, 2, 3 or 4 substituentscomprising reacting a phenyl halide of the formula (II) with a pyrazole derivative of the formula (III) in whichX is chlorine, iodine or bromine; andR, n, R, m and A are each as defined above,in the presence of a base and a catalytic system comprising a ligand and a metal compound selected from palladium compounds, iron compounds and copper compounds.

Process for preparing 1-phenylpyrazoles

Process using grignard reagents

The present invention relates to N-carbomethoxy-N-methoxy-(2-chloromethyl)-aniline compounds of the formula I, wherein: n is 0, 1, 2 or 3, each Ris independently selected from halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy or C1-C4-haloalkoxy. The invention also relates to processes and intermediates for preparing such compounds of formula I. The invention furthermore relates to processes for preparing 2-(pyrazol-3'-yloxymethylene)-anilides in which compounds of formula I are applied as precursors. 

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Mannheim, Germany

Maximilian Dochnahl