Nihon Nohyaku Co., Ltd.

Taisho Pharmaceutical Co., Ltd.

National Institute of Radiological Sciences

Makoto Goto

Shinsuke Fujioka

Masanori Tohnishi

Masayuki Morimoto

Hayami Nakao

Minoru Yamaguchi

Atsuro Nakazato

Takashi Furuya

Tetsuya Suhara

Hiroto Harayama

Ming-Rong Zhang

Kazutoshi Suzuki

The present invention provides a substituted anilide derivative of formula (I): {wherein Z is a group of formula (II) or (III) (in these formulas, A is C-Calkylene, C-Calkenylene, etc., Ris H, halogen, &#x2014;C(R)&#x2550;NOR, (substituted) phenyl, (substituted) heterocyclic ring, -A-R, etc.; Ris H, C-Calkyl, etc.), Ris H, C-Calkyl, etc.; Ris H, F, fluoro C-Calkyl; Rf is F, fluoro C-Calkyl; 1 is 0 to 2; Y is halogen, (substituted) phenyl, (substituted) phenoxy, etc.; and m is 0 to 3}, an intermediate thereof, an agrohorticultural agent, and a method for the use thereof. The compound of the present invention exhibits, at a low dosage, high uptake and translocation from the root and an excellent insecticidal effect especially when applied to soil.

Substituted aromatic amide derivative, intermediate thereof, agrohorticultural insecticide containing thereof and method for the use thereof

Sulfonamide derivatives represented by general formula (I) or salts thereof; insecticides for agricultural and horticultural use containing the same as the active ingredient; and usage thereof: [wherein A is optionally substituted (C&#x2013;C)alkylene, (C&#x2013;C)alkenylene or the like; Ris H, optionally substituted (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl, (C&#x2013;C)cycloalkyl or the like; R, Rand Rare each H, (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl or the like, or Rand A or Rand Rmay form a 3- to 8-membered ring which may be interrupted by one to three atoms selected from among O, S and N; Q is C or N; X and Y are each halogen, CN, NO, (C&#x2013;C)alkyl, (C&#x2013;C)alkenyl or the like; m is 0 to 2; n is 0 to 3; and two adjacent Xs or Ys on the aromatic ring may be united to form a fused ring]. The compounds exhibit excellent insecticidal activity against insect pests resistant to existing pesticides even when applied in dosages lower than those of similar pesticides.

Sulfonamide derivatives, insecticides for agricultural and horticultural use, and usage thereof

A phenyloxyaniline derivative useful as a ligand for peripheral benzodiazepine receptor having a strong affinity and a high selectivity, which is represented by formula (1):wherein Xand Xare same or different and each is hydrogen atom or halogen atom; Rand Rare same or different and each is hydrogen atom, an alkyl group having 1 to 10 carbon(s) or a halogen-substituted alkyl group having 1 to 10 carbon(s); and Ris a halogen-substituted alkyl group having 1 to 5 carbon(s), or a radioisotope thereof.

Phenyloxyaniline derivatives

Growing community of inventors

Yokohama, Japan

Makoto Goto