Ube Industries, Inc.

Sankyo Company, Limited

Rikagaku Kenkyusho

The Institute of Physical and Chemical Research

Katsutoshi Fujii

Tokio Obata

Shoji Shikita

Mikio Kojima

Takeo Honda

Kiyoshi Tsutsumiuchi

Shigeki Nagai

Takashi Kobayashi

Kiroku Oda

Shinji Yokoi

Yasuhisa Fukuda

Yoshinori Yamanaka

Kazuto Nakagami

Akira Ooka

Hirosuke Yoshioka

Haruo Yoshiya

Shinsaku Kobayashi

Kenji Nishimura

Yuji Akiyoshi

Toshinobu Tanaka

Katsuo Kamoshita

Isamu Narita

Ryuji Kobayashi

Hideakira Tsuji

Keigo Matsumoto

Shinjiro Yamamoto

Isao Nakayama

Toshiharu Kamioka

Yasushi Nakamoto

Shin Suizu

Kouichi Goka

Youichi Yoshida

Kiyashi Tsutsumiuchi

Tatsumi Tanaka

Koji Hatano

Kenji Nishimura, Deceased

The present invention relates to a 6-(1-fluoroethyl)-5-iodo-4-aminopyrimidine compound represented by the following formula (1):

6-(1-fluoroethyl)-5-iodo-4-aminopyrimidine compounds process for preparation of the same and pest controllers for agricultural and horticultural use

5-Iodo-4-phenethylaminopyrimidine derivative, intermediate thereof, processes for producing the same and agricultural and horticultural pesticides

N-[(fluoroalkoxy) phenoxyalkyl]benzamide compounds, intermediates

Disclosed are an oxazoline compound represented by the formula (I): ##STR1## wherein R.sup.1 represents halogen, hydrogen, alkyl, alkoxy, haloalkyl, haloalkoxy, phenyl, phenoxy, benzyl, benzyloxy, pyridyloxy, pyridylmethyloxy, alkoxy-substituted alkyl, nitro, cyanomethyloxy, haloalkylsulfonyloxy, alkylsulfonyloxy, or alkylthio; R.sup.2 represents hydrogen, halogen, alkyl, haloalkyl, alkoxy, alkylthio, or haloalkoxy; R.sup.1 and R.sup.2 may be combined to form a saturated or unsaturated 6-membered ring with oxygen; R.sup.3 represents hydrogen, halogen or alkoxy; R.sup.4 represents hydrogen, alkyl, or halogen; R.sup.5 represents hydrogen, halogen, or alkyl; X.sup.1 represents halogen, alkyl, haloalkyl, or alkoxy; X.sup.2 represents halogen, hydrogen, or alkoxy; X.sup.3 represents hydrogen or halogen; and n represents an integer of 2 to 5; an amidoethyl halide derivative used for synthesis of the same, a process for preparing the same, and an agricultural and horticultural chemical for controlling noxious organisms comprising the same as an active ingredient.

Oxazoline derivative, process for preparing the same and agricultural

Disclosed are a 4-phenethylaminopyrimidine compound represented by the formula (I): ##STR1## wherein R.sup.1 represents halogen, hydroxyl, acyloxy, alkoxy, haloalkoxy, alkylthio, benzyloxycarbonyloxy, alkyloxycarbonyloxy, alkylsulfonyloxy, tri(alkyl)silyloxy or alkyloxycarbonylalkyloxy;

4-phenethylaminopyrimidine derivative, and agricultural and

Disclosed are a phenoxyalkylamine compound represented by the formula (I): ##STR1## wherein R.sup.1 is C.sub.1-8 alkyl group, C.sub.3-8 cycloalkyl group, a hydrogen atom, a phenyl group, or C.sub.1-4 haloalkyl group; R.sup.2 is a halogen atom, a hydrogen atom, C.sub.1-4 alkyl group, C.sub.1-4 alkoxy group or a nitro group; R.sup.1 and R.sup.2 may be linked with each other and condensed to a pyrazole ring to form a saturated 4- to 8-membered ring; R.sup.3 is C.sub.1-15 alkyl group, C.sub.3-8 cycloalkyl group, a phenyl group, C.sub.1-4 haloalkyl group, C.sub.2-8 alkoxyalkyl group, C.sub.3-6 alkenyl group, a pyridyl group, a benzyl group, C.sub.3-8 alkoxycarbonylalkyl group, a pyrazole group, or C.sub.1-4 alkoxy group; R.sup.4 is C.sub.1-4 alkyl group, a hydrogen atom or a halogen atom; R.sup.5 is C.sub.1-20 alkyl group, a hydrogen atom, C.sub.3-6 alkenyl group, a benzyl group, a phenoxy group, a halogen atom, a cyanomethyl group or --A--O--R.sup.7 where A is C.sub.1-4 alkylene group and R.sup.7 is C.sub.1-6 alkyl group, C.sub.3-6 alkenyl group, C.sub.3-6 alkynyl group or C.sub.2-5 acyl group; and R.sup.6 is a hydrogen atom, C.sub.1-4 alkyl group or a halogen atom, a process for preparing the same and a chemical for controlling noxious organisms containing the same as an effective ingredient.

Phenoxyalkylamine derivative and agricultural and horticultural chemical

Disclosed are a polyfluorinated thiazoline compound represented by the following formula (I): ##STR1## wherein Q represents a phenyl group; a phenyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; a pyridyl group; or a pyridyl group substituted by a halogen atom, a halo-lower alkyl group, a nitro group, a cyano group, a formyl group, a lower alkoxycarbonyl group or a benzoyl group; and

Polyfluorinated thiazoline derivative and chemical for controlling

Disclosed are an aralkylaminopyrimidine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a halogen atom, a lower acyloxy group, a hydroxyl group, a lower alkoxy group or a lower alkylthio group; R.sup.2 represents a lower alkyl group, a hydrogen atom or a cycloalkyl group; R.sup.3 may be the same or different and represents a lower haloalkoxy group, a hydrogen atom, a lower alkyl group, a lower alkoxy group, a halogen atom, a lower alkylthio group, a nitro group, a lower haloalkyl group, a lower alkylsulfinyl group, a lower alkylsulfonyl group, a lower haloalkylthio group or a hydroxyl group; a carbon atom to which * is attached represents an asymmetric carbon atom provided that the case where R.sup.2 is a hydrogen atom is excluded; and n represents an integer of 1 to 5. a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

Aralkylaminopyrimidine derivative, and chemical for controlling noxious

Disclosed are a novel phenoxyalkylamine compound represented by the following formula: ##STR1## wherein R.sup.1 represents a lower alkyl group or a lower haloalkyl group; R.sup.2 represents hydrogen atom or a lower alkyl group; R.sup.3 represents hydrogen atom, a lower alkyl group or a halogen atom; R.sup.4 represents a lower alkenyl group or --S--O--R.sup.6 where A represents a lower alkylene group and R.sup.6 represents a lower alkyl group, a lower alkenyl group or a lower alkynyl group; R.sup.5 represents hydrogen atom, a lower alkyl group or a halogen atom, a method for preparing the same and a chemical for controlling noxious organisms which contains the same as an active ingredient.

Phenoxyalkylamine derivative and method for controlling noxious

Disclosed are a thiazoline compound represented by the following formula (I): ##STR1## wherein R represents hydrogen atom or a lower alkyl group, X represents oxygen atom or sulfur atom, and Q represents Ar (where Ar represents a substituted or unsubstituted phenyl group or a substituted or unsubstituted naphthyl group) or ##STR2## (where Y represents a halogen atom, a lower alkyl group, a lower alkoxy group, a lower haloalkyl group, a lower haloalkoxy group, nitro group, acetyl group or cyano group and n represents an integer of 0 to 5), a process for preparing the same and a chemical for controlling noxious organisms containing the same as an active ingredient.

Thiazoline derivative, process for preparing the same and chemical for

Disclosed are a compound of the formula (I) or an acid addition salt thereof: ##STR1## wherein Q represents R.sup.1 , R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, n and z are defined as in the specification, preparation method thereof and fungicides containing the same.

Aralkylamine derivatives, and fungicides containing the same

An aminopyrimidine compound of the formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, an alkyl group, a cycloalkyl group or a halogen atom;

Aminopyrimidine derivatives and harmful organisms preventive agent

A compound represented by the formula: ##STR1## wherein R.sub.1 represents hydrogen atom, a halogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.2 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; R.sub.3 represents an alkyl group having 1 to 8 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or an aralkyl group which may be also substituted; R.sub.4 represents hydrogen atom or an alkyl group having 1 to 5 carbon atoms; n represents an integer of 4 and when R.sub.2 is an alkyl group, n represents an integer of 1 to 3; A represents an alkylene group having 1 to 5 carbon atoms; and X represents an oxygen atom or a sulfur atom and an insecticide, acaricide or fungicide comprising a compound of the formula (I) as the active ingredient.

Pyrazoleoxime derivative and insecticide, acaricide and fungicide

Disclosed are an aminopyrimidine compound or an acid addition salt thereof represented by the formula: ##STR1## wherein R1, R2, R3, R4, R5 and Y have the same meanings defined in the specification; a process for preparing the compound and insecticide or bactericide containing the compound.

Aminopyrimidine derivative and insecticide or bactericide containing the

There are disclosed a phenoxyalkylamine derivative represented by the formula: ##STR1## wherein A.sup.1 represents an alkylene group having 2 to 5 carbon atoms, R.sup.1 and R.sup.2 each represent hydrogen atom or a lower alkyl group having 1 to 5 carbon atoms, R.sup.3, R.sup.4 and R.sup.5 each represent hydrogen atom, an alkyl group having 1 to 5 carbon atoms or a halogen atom, R.sup.6 represents hydrogen atom, an alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms or a group --A.sup.2 --X--R.sup.7, A.sup.2 represents an alkylene group having 1 to 5 carbon atoms, X represents oxygen atom or sulfur atom, R.sup.7 represents a lower alkyl group having 1 to 5 carbon atoms, an alkenyl group having 3 to 5 carbon atoms, an alkynyl group having 3 to 5 carbon atoms or a substituted or unsubstituted aralkyl group, and an insecticide, an acaricide and a fungicide for agriculture and horticulture, which comprises a carrier and the above phenoxyalkylamine derivative represented as the active ingredient.

Phenoxyalkylamine derivatives, and insecticides, acaricides and

Growing community of inventors

Ube, Japan

Katsutoshi Fujii